Beta-1 adrenergic receptor — Drug Target
All drugs that target Beta-1 adrenergic receptor — marketed and clinical-stage. Includes 24 drug classes acting on this target.
Drug classes
Beta-1 selective adrenergic antagonist (beta-blocker) · Beta-1 selective adrenergic receptor antagonist (cardioselective beta-blocker) · bevantolol · beta-Adrenergic Blocker [EPC] · beta-Adrenergic Blocker · etilefrine · bretylium · beta blocker · celiprolol · Beta-1 selective adrenergic antagonist (beta blocker) · Beta-1 selective adrenergic receptor antagonist · arbutamine
Marketed (30)
- Atenolol Pill · Tartu University Hospital · Beta-1 selective adrenergic antagonist (beta-blocker) · Cardiovascular
Atenolol is a beta-1 selective adrenergic receptor antagonist that reduces heart rate and blood pressure by blocking the effects of norepinephrine and epinephrine on the heart. - Bisoprolol versus Nebivolol · Clinical Hospital Center Zemun · Beta-1 selective adrenergic receptor antagonist (cardioselective beta-blocker) · Cardiovascular
Both bisoprolol and nebivolol are beta-1 selective adrenergic receptor antagonists that reduce heart rate and blood pressure by blocking sympathetic nervous system signaling in the heart. - Atenolol Succinate Oral Tablet · Damanhour Teaching Hospital · Beta-1 selective adrenergic antagonist (beta-blocker) · Cardiovascular
Atenolol succinate is a beta-1 selective adrenergic receptor antagonist that reduces heart rate and blood pressure by blocking the effects of catecholamines on the heart. - Calvan · bevantolol · Cardiovascular
- Low Dose Bisoprolol · Merck KGaA, Darmstadt, Germany · Beta-1 selective adrenergic antagonist (beta-blocker) · Cardiovascular
Bisoprolol is a beta-1 selective adrenergic receptor antagonist that reduces heart rate and blood pressure by blocking the effects of catecholamines on the heart. - Metoprolole (Selo-Zok ®) · Rigshospitalet, Denmark · Beta-1 selective adrenergic antagonist (beta-blocker) · Cardiovascular
Metoprolol is a selective beta-1 adrenergic receptor antagonist that reduces heart rate and blood pressure by blocking the effects of norepinephrine and epinephrine on the heart. - Visken · beta-Adrenergic Blocker [EPC] · Cardiovascular
- Normodyne · Merck & Co. · beta-Adrenergic Blocker · Cardiovascular
- Etilefrin · etilefrine · Cardiovascular
- Different doses of Metoprolol. · Xiangya Hospital of Central South University · Beta-1 selective adrenergic antagonist (beta-blocker) · Cardiovascular
Metoprolol is a selective beta-1 adrenergic receptor antagonist that reduces heart rate, blood pressure, and cardiac workload. - Bretylium Tosylate · Pfizer · bretylium · Neuroscience
- Brevibloc In Plastic Container · Pfizer · beta-Adrenergic Blocker · Cardiovascular
Brevibloc works by blocking the beta-1 adrenergic receptor, which reduces the heart's response to stress and increases heart rate. - Baracle Tab.® · Seoul St. Mary's Hospital · beta blocker · Cardiovascular
Baracle Tab. is a beta blocker used to treat hypertension and prevent myocardial infarction. - Selectol · celiprolol · Cardiovascular
- Prophylactic esmolol · Hospital de Base · Beta-1 selective adrenergic antagonist (beta blocker) · Cardiovascular / Perioperative Medicine
Esmolol is a selective beta-1 adrenergic receptor antagonist that rapidly reduces heart rate and blood pressure to prevent perioperative tachycardia and hypertension. - Nebivolol (NEB) · Mylan Bertek Pharmaceuticals · Beta-1 selective adrenergic receptor antagonist · Cardiovascular
Nebivolol is a selective beta-1 adrenergic receptor antagonist that also has vasodilatory properties through nitric oxide release. - Sectral · Promius Pharma · beta-Adrenergic Blocker · Neuroscience
- Optipranolol · Bausch Health · beta-Adrenergic Blocker · Cardiovascular
- Ocupress · beta-Adrenergic Blocker · Cardiovascular
- Genesa · arbutamine · Cardiovascular
- High Dose Bisoprolol · Merck KGaA, Darmstadt, Germany · Beta-1 selective adrenergic receptor antagonist (beta-blocker) · Cardiovascular
High-dose bisoprolol is a selective beta-1 adrenergic receptor antagonist that reduces heart rate and cardiac contractility to lower blood pressure and improve cardiac function. - Nebivolol Pill · Tartu University Hospital · Beta-1 selective adrenergic antagonist (beta-blocker) · Cardiovascular
Nebivolol is a selective beta-1 adrenergic receptor antagonist that reduces heart rate and blood pressure while preserving vasodilatory properties through nitric oxide release. - Metoprolol (MET) · Tel-Aviv Sourasky Medical Center · Beta-1 selective adrenergic receptor antagonist (beta-blocker) · Cardiovascular
Metoprolol is a beta-1 selective adrenergic receptor antagonist that reduces heart rate, blood pressure, and cardiac workload. - Onoact · Aop Hlth Us · landiolol · Cardiovascular
Onoact works by blocking the beta-1 adrenergic receptor, which helps to slow down abnormal heart rhythms. - Betaxon · Alcon Pharms Ltd · levobetaxolol · Cardiovascular
- Zebeta · Teva · beta-Adrenergic Blocker · Cardiovascular
- Betoptic · Novartis · beta-Adrenergic Blocker · Cardiovascular
Betaxolol works by blocking the beta-1 adrenergic receptor in the heart and eyes, reducing heart rate and pressure, and decreasing intraocular pressure. - Nebivolol Tablets · Ain Shams University · Beta-1 selective adrenergic receptor antagonist (beta-blocker) · Cardiovascular
Nebivolol is a selective beta-1 adrenergic receptor antagonist that reduces heart rate and blood pressure while also promoting nitric oxide-mediated vasodilation. - Post-CPB Drug: Dobutamine Hydrochloride · University Health Network, Toronto · Beta-1 adrenergic agonist · Cardiovascular
Dobutamine is a beta-1 adrenergic agonist that increases cardiac contractility and heart rate to improve cardiac output in patients with low cardiac function. - brand name metoprolol ER · University of Florida · Beta-1 selective adrenergic receptor antagonist (beta-blocker) · Cardiovascular
Metoprolol ER is a beta-1 selective adrenergic receptor antagonist that reduces heart rate and blood pressure by blocking the effects of norepinephrine and epinephrine on the heart.
Phase 3 pipeline (10)
- Landiolol HCl · Medical University of Vienna · Beta-1 selective adrenergic antagonist (beta-blocker) · Cardiovascular
Landiolol HCl is an ultra-short-acting beta-1 selective adrenergic antagonist that rapidly reduces heart rate and cardiac workload. - Levobetaxolol eye drops · Zhaoke (Guangzhou) Ophthalmology Pharmaceutical Ltd. · Selective beta-1 adrenergic antagonist (beta-blocker) · Ophthalmology
Levobetaxolol is a selective beta-1 adrenergic receptor antagonist that reduces intraocular pressure by decreasing aqueous humor production in the eye. - metoprolol/HCT · Abbott · Beta-blocker · Cardiovascular
Metoprolol/HCT is a beta-blocker that works by blocking the effects of the hormone epinephrine, and also has a diuretic effect to reduce blood pressure. - Esmolol Injection [Brevibloc] · Consorcio Centro de Investigación Biomédica en Red (CIBER) · Beta-1 selective adrenergic antagonist · Cardiovascular
Esmolol is a selective beta-1 adrenergic receptor antagonist that rapidly blocks sympathetic stimulation of the heart, reducing heart rate and blood pressure. - Sustained-release Metoprolol Succinate · Jiangsu HengRui Medicine Co., Ltd. · Beta-blocker · Cardiovascular
Metoprolol succinate is a beta-blocker that works by blocking the effects of the hormone epinephrine, also known as adrenaline, and slowing the heart rate and reducing its workload. - DOBUTamine Injectable Solution · The Young Investigator Group of Cardiovascular Research · Beta-1 adrenergic agonist · Cardiovascular
Dobutamine is a beta-1 adrenergic agonist that increases cardiac contractility and heart rate to improve cardiac output. - Seloken ZOK/Toprol-XL · AstraZeneca · beta-blocker · Cardiovascular
Seloken ZOK/Toprol-XL is a beta-blocker that works by blocking the effects of the hormone epinephrine, also known as adrenaline, and slowing the heart rate and reducing its workload. - Nebivolol and Atenolol · Mylan Bertek Pharmaceuticals · Beta-blocker (beta-1 selective adrenergic antagonist) · Cardiovascular
Nebivolol and atenolol are beta-blockers that reduce heart rate and blood pressure by blocking beta-adrenergic receptors on the heart and blood vessels. - cardio-selective beta blocker group · Sherief Abd-Elsalam · Cardio-selective beta blocker · Cardiovascular
Blocks beta-1 adrenergic receptors to reduce heart rate and blood pressure. - Betaxolol eye drops · Zhaoke (Guangzhou) Ophthalmology Pharmaceutical Ltd. · Selective beta-1 adrenergic antagonist (beta-blocker) · Ophthalmology
Betaxolol is a selective beta-1 adrenergic receptor antagonist that reduces intraocular pressure by decreasing aqueous humor production in the eye.
Phase 2 pipeline (3)
- Esmolol administration · Assistance Publique - Hôpitaux de Paris · Beta blocker · Cardiovascular
Beta-1 adrenergic receptor antagonist - ETILEFRINE PIVALATE · etilefrine pivalate · Cardiovascular
Etilefrine pivalate works by stimulating the beta-1 adrenergic receptor to increase heart rate and contractility. - LEVDOBUTAMINE · Cardiovascular
Levodobutamine works by binding to and activating the beta-1 adrenergic receptor, which plays a key role in regulating heart function.