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Esmolol administration

Assistance Publique - Hôpitaux de Paris · Phase 2 active Small molecule

Beta-1 adrenergic receptor antagonist

Beta-1 adrenergic receptor antagonist Used for Hypertension, Tachyarrhythmias.

At a glance

Generic nameEsmolol administration
Also known asBREVIBLOC 10 mg/ml, Drug by Qilu Pharmaceutical Co, Shandong, China
SponsorAssistance Publique - Hôpitaux de Paris
Drug classBeta blocker
TargetBeta-1 adrenergic receptor
ModalitySmall molecule
Therapeutic areaCardiovascular
PhasePhase 2

Mechanism of action

Esmolol is a selective beta-1 adrenergic receptor antagonist that reduces heart rate and blood pressure.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results