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Levobetaxolol eye drops

Zhaoke (Guangzhou) Ophthalmology Pharmaceutical Ltd. · Phase 3 active Small molecule

Levobetaxolol is a selective beta-1 adrenergic receptor antagonist that reduces intraocular pressure by decreasing aqueous humor production in the eye.

Levobetaxolol is a selective beta-1 adrenergic receptor antagonist that reduces intraocular pressure by decreasing aqueous humor production in the eye. Used for Glaucoma, Ocular hypertension.

At a glance

Generic nameLevobetaxolol eye drops
SponsorZhaoke (Guangzhou) Ophthalmology Pharmaceutical Ltd.
Drug classSelective beta-1 adrenergic antagonist (beta-blocker)
TargetBeta-1 adrenergic receptor
ModalitySmall molecule
Therapeutic areaOphthalmology
PhasePhase 3

Mechanism of action

As a beta-blocker, levobetaxolol selectively inhibits beta-1 adrenergic receptors in the ciliary body of the eye, which reduces the production and secretion of aqueous humor. This decrease in aqueous humor production leads to lower intraocular pressure, making it effective for treating glaucoma and ocular hypertension. The selective beta-1 activity minimizes systemic side effects compared to non-selective beta-blockers.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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