What drugs target Histamine H2 receptor?

10+ drugs target Histamine H2 receptor, including Bentyl, Ebrodin, Histalog, Tagamet, Famotidine (FAM).

What drug classes act on Histamine H2 receptor?

Drug classes acting on Histamine H2 receptor include Anticholinergic, ebrotidine, betazole, Histamine-2 Receptor Antagonist [EPC], H2-receptor antagonist.

Histamine H2 receptor — Drug Target

10 drugs 7 marketed 2 in Phase 3

All drugs that target Histamine H2 receptor — marketed and clinical-stage. Includes 7 drug classes acting on this target.

Drug classes

Anticholinergic · ebrotidine · betazole · Histamine-2 Receptor Antagonist [EPC] · H2-receptor antagonist · H2 receptor antagonist · niperotidine

Marketed (7)

Bentyl · Forest Labs Inc · Anticholinergic · Neuroscience
Ebrodin · ebrotidine · Cardiovascular
Histalog · betazole · Other
Tagamet · Histamine-2 Receptor Antagonist [EPC] · Cardiovascular
Famotidine (FAM) · Bristol-Myers Squibb · H2-receptor antagonist · Gastroenterology
Famotidine is a histamine H2-receptor antagonist that reduces gastric acid secretion by blocking histamine-mediated stimulation of parietal cells in the stomach.
Axid Ar · Histamine-2 Receptor Antagonist [EPC] · Cardiovascular
Drug: cimetidine · University of Maryland, Baltimore · H2 receptor antagonist · Gastroenterology
Cimetidine blocks histamine H2 receptors on gastric parietal cells to reduce stomach acid production.

Phase 3 pipeline (2)

H2 Receptor Antagonist · Merck Sharp & Dohme LLC · H2 receptor antagonist · Gastroenterology
H2 receptor antagonists block histamine H2 receptors on gastric parietal cells to reduce stomach acid secretion.
Cimetidine IV · Bausch Health Americas, Inc. · H2-receptor antagonist · Gastroenterology
Cimetidine is a histamine H2-receptor antagonist that reduces gastric acid secretion by blocking histamine-mediated stimulation of parietal cells.

Phase 2 pipeline (1)

Perultid · niperotidine · Other
Perultid works by blocking histamine receptors in the stomach to reduce acid production.