GnRH antagonist
This page covers all GnRH antagonist drugs tracked by Drug Landscape: marketed products and active clinical-stage compounds, targeting GnRH receptor, GnRH receptor (GnRHR).
Targets
GnRH receptor · GnRH receptor (GnRHR)
Marketed (6)
- Antagon ™ · EMD Serono · Reproductive Medicine / Fertility
Antagon is a gonadotropin-releasing hormone (GnRH) antagonist that rapidly suppresses luteinizing hormone (LH) and follicle-stimulating hormone (FSH) to prevent premature ovulation during assisted reproductive technology. - cetrorelix (cetrotide) · Eugonia · Reproductive/Fertility
Cetrorelix is a gonadotropin-releasing hormone (GnRH) antagonist that blocks GnRH receptors to suppress luteinizing hormone (LH) and follicle-stimulating hormone (FSH) secretion. - Antagonist GnRH Cetrotide · Instituto Valenciano de Infertilidad, IVI VALENCIA · Reproductive Medicine / Fertility
Cetrotide is a GnRH antagonist that directly blocks gonadotropin-releasing hormone receptors to suppress luteinizing hormone and follicle-stimulating hormone secretion. - Ganirelix Acetate, Cetrolix Acetate · Assaf-Harofeh Medical Center · Reproductive Medicine / Fertility
Ganirelix and Cetrolix are gonadotropin-releasing hormone (GnRH) antagonists that block GnRH receptors to suppress luteinizing hormone (LH) and follicle-stimulating hormone (FSH) secretion. - GnRH antagonist-Cetrorelix · University of Edinburgh · Reproductive Medicine / Endocrinology
Cetrorelix blocks gonadotropin-releasing hormone (GnRH) receptors to suppress luteinizing hormone and follicle-stimulating hormone secretion. - Degarelix (LHRH antagonist) · Rabin Medical Center · Oncology
Degarelix is a gonadotropin-releasing hormone (GnRH) antagonist that rapidly suppresses luteinizing hormone and follicle-stimulating hormone, leading to testosterone suppression.
Phase 3 pipeline (8)
- Ganirelix (GnRH antagonist) · Instituto Valenciano de Infertilidad, IVI VALENCIA · Reproductive Medicine / Fertility
Ganirelix blocks gonadotropin-releasing hormone (GnRH) receptors to suppress luteinizing hormone (LH) and prevent premature ovulation during assisted reproductive procedures. - SHR7280 simulant； Ganirelix Acetate Injection · Jiangsu HengRui Medicine Co., Ltd. · Reproductive Medicine / Fertility
Ganirelix acetate is a gonadotropin-releasing hormone (GnRH) antagonist that suppresses luteinizing hormone (LH) and follicle-stimulating hormone (FSH) secretion. - Cetrorelix 78+78 · AEterna Zentaris · Oncology; Reproductive/Endocrinology
Cetrorelix is a gonadotropin-releasing hormone (GnRH) antagonist that suppresses luteinizing hormone and follicle-stimulating hormone to inhibit ovarian steroid production. - Cetrorelix Pamoate · AEterna Zentaris · Oncology; Reproductive Health
Cetrorelix pamoate is a gonadotropin-releasing hormone (GnRH) antagonist that blocks GnRH receptors to suppress luteinizing hormone and follicle-stimulating hormone secretion. - Cetrotide Injectable Product · El Shatby University Hospital for Obstetrics and Gynecology · Reproductive/Fertility
Cetrotide is a gonadotropin-releasing hormone (GnRH) antagonist that blocks GnRH receptors to suppress luteinizing hormone and follicle-stimulating hormone secretion. - Relugolix Combination Therapy · Sumitomo Pharma Switzerland GmbH · Oncology
Relugolix is a gonadotropin-releasing hormone (GnRH) antagonist that suppresses luteinizing hormone and follicle-stimulating hormone, leading to rapid reduction of testosterone and estrogen levels. - SHR7280；Ganirelix Acetate Injection simulant · Jiangsu HengRui Medicine Co., Ltd. · Reproductive/Fertility
Ganirelix acetate is a gonadotropin-releasing hormone (GnRH) antagonist that suppresses luteinizing hormone (LH) and follicle-stimulating hormone (FSH) secretion. - Ganirelix 0.25 mg. · Instituto de Investigacion Sanitaria La Fe · Reproductive Medicine / Fertility
Ganirelix is a gonadotropin-releasing hormone (GnRH) antagonist that suppresses luteinizing hormone (LH) and follicle-stimulating hormone (FSH) secretion to prevent premature ovulation during assisted reproductive procedures.
Phase 2 pipeline (1)
- Analogous GnRH antagonist · Merck KGaA, Darmstadt, Germany · Oncology; Reproductive/Endocrinology
This GnRH antagonist blocks gonadotropin-releasing hormone receptors to suppress luteinizing hormone and follicle-stimulating hormone, reducing sex hormone production.