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TIVA - Neostigmine 70

Pontificia Universidade Catolica de Sao Paulo · FDA-approved active Small molecule

TIVA - Neostigmine 70 is a Acetylcholinesterase inhibitor Small molecule drug developed by Pontificia Universidade Catolica de Sao Paulo. It is currently FDA-approved for Reversal of neuromuscular blockade, Myasthenia gravis, Postoperative ileus and urinary retention. Also known as: TIVA.

Neostigmine is a reversible acetylcholinesterase inhibitor that increases acetylcholine levels at the neuromuscular junction and in the central nervous system.

Neostigmine is a reversible acetylcholinesterase inhibitor that increases acetylcholine levels at the neuromuscular junction and in the central nervous system. Used for Reversal of neuromuscular blockade, Myasthenia gravis, Postoperative ileus and urinary retention.

At a glance

Generic nameTIVA - Neostigmine 70
Also known asTIVA
SponsorPontificia Universidade Catolica de Sao Paulo
Drug classAcetylcholinesterase inhibitor
TargetAcetylcholinesterase
ModalitySmall molecule
Therapeutic areaNeurology
PhaseFDA-approved

Mechanism of action

By inhibiting the enzyme acetylcholinesterase, neostigmine prevents the breakdown of acetylcholine, leading to increased acetylcholine concentration in synaptic spaces. This enhances cholinergic neurotransmission at the neuromuscular junction and autonomic nervous system sites. The drug is used to reverse neuromuscular blockade and treat myasthenia gravis by prolonging the action of available acetylcholine.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about TIVA - Neostigmine 70

What is TIVA - Neostigmine 70?

TIVA - Neostigmine 70 is a Acetylcholinesterase inhibitor drug developed by Pontificia Universidade Catolica de Sao Paulo, indicated for Reversal of neuromuscular blockade, Myasthenia gravis, Postoperative ileus and urinary retention.

How does TIVA - Neostigmine 70 work?

Neostigmine is a reversible acetylcholinesterase inhibitor that increases acetylcholine levels at the neuromuscular junction and in the central nervous system.

What is TIVA - Neostigmine 70 used for?

TIVA - Neostigmine 70 is indicated for Reversal of neuromuscular blockade, Myasthenia gravis, Postoperative ileus and urinary retention.

Who makes TIVA - Neostigmine 70?

TIVA - Neostigmine 70 is developed and marketed by Pontificia Universidade Catolica de Sao Paulo (see full Pontificia Universidade Catolica de Sao Paulo pipeline at /company/pontificia-universidade-catolica-de-sao-paulo).

Is TIVA - Neostigmine 70 also known as anything else?

TIVA - Neostigmine 70 is also known as TIVA.

What drug class is TIVA - Neostigmine 70 in?

TIVA - Neostigmine 70 belongs to the Acetylcholinesterase inhibitor class. See all Acetylcholinesterase inhibitor drugs at /class/acetylcholinesterase-inhibitor.

What development phase is TIVA - Neostigmine 70 in?

TIVA - Neostigmine 70 is FDA-approved (marketed).

What are the side effects of TIVA - Neostigmine 70?

Common side effects of TIVA - Neostigmine 70 include Increased salivation, Bronchospasm, Bradycardia, Muscle fasciculations, Nausea and vomiting.

What does TIVA - Neostigmine 70 target?

TIVA - Neostigmine 70 targets Acetylcholinesterase and is a Acetylcholinesterase inhibitor.

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