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Ondansetron oral tablets
Ondansetron oral tablets is a Serotonin 5-HT3 receptor antagonist Small molecule drug developed by GlaxoSmithKline. It is currently in Phase 3 development for Prevention of nausea and vomiting caused by cancer chemotherapy, Prevention of nausea and vomiting caused by radiation therapy. Also known as: Dexamethasone intravenous, Casopitant (GW679769) oral tablets, Casopitant (GW679769) intravenous.
Ondansetron works by blocking serotonin receptors in the body, which helps to reduce nausea and vomiting.
Ondansetron works by blocking serotonin receptors in the body, which helps to reduce nausea and vomiting. Used for Prevention of nausea and vomiting caused by cancer chemotherapy, Prevention of nausea and vomiting caused by radiation therapy.
At a glance
| Generic name | Ondansetron oral tablets |
|---|---|
| Also known as | Dexamethasone intravenous, Casopitant (GW679769) oral tablets, Casopitant (GW679769) intravenous |
| Sponsor | GlaxoSmithKline |
| Drug class | Serotonin 5-HT3 receptor antagonist |
| Target | 5-HT3 receptor |
| Modality | Small molecule |
| Therapeutic area | Oncology |
| Phase | Phase 3 |
Mechanism of action
This is achieved through the antagonism of 5-HT3 receptors in the central nervous system and the gastrointestinal tract. By blocking these receptors, ondansetron reduces the vomiting reflex and alleviates nausea.
Approved indications
- Prevention of nausea and vomiting caused by cancer chemotherapy
- Prevention of nausea and vomiting caused by radiation therapy
Common side effects
- Headache
- Dizziness
- Constipation
- Diarrhea
- Fatigue
Key clinical trials
- Phase I PK and Safety Study of Ondansetron Inhalation Powder (PHASE1)
- The Efficacy and Safety of Liposomal Bupivacaine for Transversus Abdominis Plane Block in Relieving Postoperative Pain After Laparoscopic Surgery (NA)
- The Efficacy and Safety of Liposomal Bupivacaine for Transversus Abdominis Plane Block in Relieving Postoperative Pain After Laparoscopic Surgery in Gynecologic Oncology (NA)
- The Efficacy and Safety of Liposomal Bupivacaine in Relieving Postoperative Pain After Laparoscopic Surgery (NA)
- Assessment of Medrol Dosepak to Reduce Opioid Consumption in Foot and Ankle Surgical Patients (PHASE2)
- The Efficacy and Safety of Liposomal Bupivacaine in Relieving Postoperative Pain After Video-assisted Thoracoscopic Surgery (NA)
- The Efficacy and Safety of Liposomal Bupivacaine in Relieving Postoperative Pain After Hemorrhoid Surgery (NA)
- The Efficacy and Safety of Liposomal Bupivacaine for Rhomboid Intercostal Nerve Block in Relieving Postoperative Pain After Video-assisted Thoracoscopic Surgery (NA)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Ondansetron oral tablets CI brief — competitive landscape report
- Ondansetron oral tablets updates RSS · CI watch RSS
- GlaxoSmithKline portfolio CI
Frequently asked questions about Ondansetron oral tablets
What is Ondansetron oral tablets?
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Related
- Drug class: All Serotonin 5-HT3 receptor antagonist drugs
- Target: All drugs targeting 5-HT3 receptor
- Manufacturer: GlaxoSmithKline — full pipeline
- Therapeutic area: All drugs in Oncology
- Indication: Drugs for Prevention of nausea and vomiting caused by cancer chemotherapy
- Indication: Drugs for Prevention of nausea and vomiting caused by radiation therapy
- Also known as: Dexamethasone intravenous, Casopitant (GW679769) oral tablets, Casopitant (GW679769) intravenous
- Compare: Ondansetron oral tablets vs similar drugs
- Pricing: Ondansetron oral tablets cost, discount & access