Last reviewed · How we verify
epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile
epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile is a anthracycline antibiotic, taxane, alkylating agent, antifolate, thymidylate synthase inhibitor Small molecule drug developed by Sanofi. It is currently in Phase 3 development for Metastatic breast cancer, Metastatic non-small cell lung cancer, Metastatic ovarian cancer.
Epidoxorubicine is an anthracycline antibiotic that intercalates DNA strands, thereby inhibiting the progression of topoisomerase II and inducing apoptosis in cancer cells. Docetaxel is a taxane that stabilizes microtubules, preventing cell division and leading to cell death. Ciclophosphamide is an alkylating agent that adds an alkyl group to DNA, causing cross-linking and DNA damage. Methotrexate is an antifolate that inhibits dihydrofolate reductase, leading to a decrease in DNA synthesis and cell proliferation. Fluorouracile is a thymidylate synthase inhibitor that disrupts DNA synthesis and repair.
Epidoxorubicine is an anthracycline antibiotic that intercalates DNA strands, thereby inhibiting the progression of topoisomerase II and inducing apoptosis in cancer cells. Docetaxel is a taxane that stabilizes microtubules, preventing cell division and leading to cell death. Ciclophosphamide is an alkylating agent that adds an alkyl group to DNA, causing cross-linking and DNA damage. Methotrexate is an antifolate that inhibits dihydrofolate reductase, leading to a decrease in DNA synthesis and cell proliferation. Fluorouracile is a thymidylate synthase inhibitor that disrupts DNA synthesis and repair. Used for Metastatic breast cancer, Metastatic non-small cell lung cancer, Metastatic ovarian cancer.
At a glance
| Generic name | epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile |
|---|---|
| Sponsor | Sanofi |
| Drug class | anthracycline antibiotic, taxane, alkylating agent, antifolate, thymidylate synthase inhibitor |
| Target | topoisomerase II, microtubules, dihydrofolate reductase, thymidylate synthase |
| Modality | Small molecule |
| Therapeutic area | Oncology |
| Phase | Phase 3 |
Mechanism of action
Epidoxorubicine's mechanism of action involves the intercalation of DNA strands, which inhibits the progression of topoisomerase II and induces apoptosis in cancer cells. Docetaxel's mechanism of action involves the stabilization of microtubules, preventing cell division and leading to cell death. Ciclophosphamide's mechanism of action involves the addition of an alkyl group to DNA, causing cross-linking and DNA damage. Methotrexate's mechanism of action involves the inhibition of dihydrofolate reductase, leading to a decrease in DNA synthesis and cell proliferation. Fluorouracile's mechanism of action involves the inhibition of thymidylate synthase, disrupting DNA synthesis and repair.
Approved indications
- Metastatic breast cancer
- Metastatic non-small cell lung cancer
- Metastatic ovarian cancer
- Metastatic pancreatic cancer
Common side effects
- Neutropenia
- Anemia
- Thrombocytopenia
- Nausea and vomiting
- Diarrhea
- Fatigue
- Mucositis
- Hair loss
Key clinical trials
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile CI brief — competitive landscape report
- epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile updates RSS · CI watch RSS
- Sanofi portfolio CI
Frequently asked questions about epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile
What is epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile?
How does epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile work?
What is epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile used for?
Who makes epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile?
What drug class is epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile in?
What development phase is epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile in?
What are the side effects of epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile?
What does epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile target?
Related
- Drug class: All anthracycline antibiotic, taxane, alkylating agent, antifolate, thymidylate synthase inhibitor drugs
- Target: All drugs targeting topoisomerase II, microtubules, dihydrofolate reductase, thymidylate synthase
- Manufacturer: Sanofi — full pipeline
- Therapeutic area: All drugs in Oncology
- Indication: Drugs for Metastatic breast cancer
- Indication: Drugs for Metastatic non-small cell lung cancer
- Indication: Drugs for Metastatic ovarian cancer
- Compare: epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile vs similar drugs
- Pricing: epidoxorubicine, docetaxel, ciclophosphamide, methotrexate, fluorouracile cost, discount & access