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Cisplatin (as radiosensitizer)
Cisplatin (as radiosensitizer) is a Platinum-based chemotherapy agent Small molecule drug developed by Merck Sharp & Dohme LLC. It is currently in Phase 3 development for Concurrent chemoradiation for locally advanced cancers (head and neck, cervical, lung, esophageal). Also known as: Platinol®, Platinol®-AQ.
Cisplatin acts as a radiosensitizer by forming DNA adducts that enhance the cytotoxic effects of ionizing radiation, making cancer cells more susceptible to radiation-induced damage.
Cisplatin acts as a radiosensitizer by forming DNA adducts that enhance the cytotoxic effects of ionizing radiation, making cancer cells more susceptible to radiation-induced damage. Used for Concurrent chemoradiation for locally advanced cancers (head and neck, cervical, lung, esophageal).
At a glance
| Generic name | Cisplatin (as radiosensitizer) |
|---|---|
| Also known as | Platinol®, Platinol®-AQ |
| Sponsor | Merck Sharp & Dohme LLC |
| Drug class | Platinum-based chemotherapy agent |
| Target | DNA |
| Modality | Small molecule |
| Therapeutic area | Oncology |
| Phase | Phase 3 |
Mechanism of action
Cisplatin is a platinum-based chemotherapy agent that binds to DNA and creates interstrand and intrastrand crosslinks. When combined with radiation therapy, these DNA lesions become more difficult for cells to repair, significantly enhancing radiation-induced cell death. This synergistic effect makes cisplatin an effective radiosensitizing agent in concurrent chemoradiation regimens.
Approved indications
- Concurrent chemoradiation for locally advanced cancers (head and neck, cervical, lung, esophageal)
Common side effects
- Nephrotoxicity
- Ototoxicity
- Nausea and vomiting
- Myelosuppression
- Peripheral neuropathy
- Electrolyte abnormalities (hypomagnesemia, hypokalemia)
Key clinical trials
- Study of Trastuzumab Deruxtecan Versus Standard of Care Chemotherapy for HER2-Expressing (IHC 3+/2+) Endometrial Cancer (PHASE3)
- Study of Pembrolizumab (MK-3475) in Combination With Adjuvant Chemotherapy With or Without Radiotherapy in Participants With Newly Diagnosed Endometrial Cancer After Surgery With Curative Intent (MK-3475-B21 / KEYNOTE-B21 / ENGOT-en11 / GOG-3053) (PHASE3)
- sEphB4-HSA With RT+Chemo or Cetux in Patients With Intermediate to High Risk LAHNSCC (PHASE1)
- AF CRT +/- Nimorazole in HNSCC (PHASE3)
- Erlotinib, Cisplatin, and Radiation Therapy in Treating Patients With Stage IB-Stage IVA Cervical Cancer (PHASE1)
- Cytochlor and Tetrahydrouridine as Radiosensitizers and Cisplatin Combined With Radiation Therapy in Treating Patients With Advanced Squamous Cell Carcinoma of the Oral Cavity (Mouth) or Oropharynx (Throat) (PHASE1)
- Cisplatin and Radiation Therapy With or Without Erlotinib Hydrochloride in Treating Patients With Stage III or Stage IV Head and Neck Cancer (PHASE2)
- Chemotherapy and Radiation Following Pancreatic Surgery (PHASE2)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Cisplatin (as radiosensitizer) CI brief — competitive landscape report
- Cisplatin (as radiosensitizer) updates RSS · CI watch RSS
- Merck Sharp & Dohme LLC portfolio CI
Frequently asked questions about Cisplatin (as radiosensitizer)
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Related
- Drug class: All Platinum-based chemotherapy agent drugs
- Target: All drugs targeting DNA
- Manufacturer: Merck Sharp & Dohme LLC — full pipeline
- Therapeutic area: All drugs in Oncology
- Indication: Drugs for Concurrent chemoradiation for locally advanced cancers (head and neck, cervical, lung, esophageal)
- Also known as: Platinol®, Platinol®-AQ
- Compare: Cisplatin (as radiosensitizer) vs similar drugs
- Pricing: Cisplatin (as radiosensitizer) cost, discount & access