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Bupivacaine hydrochloride 1%
Bupivacaine hydrochloride 1% is a Local anesthetic Small molecule drug developed by Express Specialty Pharmacy. It is currently in Phase 2 development for Local anesthesia. Also known as: Bupivacaine hydrochloride.
Local anesthetic by blocking sodium channels
Local anesthetic by blocking sodium channels Used for Local anesthesia.
At a glance
| Generic name | Bupivacaine hydrochloride 1% |
|---|---|
| Also known as | Bupivacaine hydrochloride |
| Sponsor | Express Specialty Pharmacy |
| Drug class | Local anesthetic |
| Target | Voltage-gated sodium channels |
| Modality | Small molecule |
| Therapeutic area | Oncology |
| Phase | Phase 2 |
Mechanism of action
Bupivacaine hydrochloride works by inhibiting the influx of sodium ions through voltage-gated sodium channels, which helps to prevent the initiation and transmission of nerve impulses.
Approved indications
- Local anesthesia
Common side effects
- Central nervous system depression
- Cardiovascular toxicity
Key clinical trials
- Arthrosemid vs. Steroid for the Management Knee Osteoarthritis (PHASE4)
- mTLIP vs QIPB for Postoperative Analgesia in Lumbar Microdiscectomy Surgery (NA)
- Continuous Epidural With Dexmedetomidine Adjuvant in Gynecologic Laparotomy (PHASE4)
- Parascapular Sub Iliocostalis Plane Block Versus Thoracic Paravertebral Plane Block for Traumatic Multiple Rib Fractures (NA)
- Intercostal Nerve Cryoablation Versus Epidural Analgesia for Nuss Repair of Pectus Excavatum (NA)
- Opioid Free and Opioid Based Anesthesia in Elective Lumbar Spine Surgery
- Comparison of Postoperative Analgesic Efficacy of Interscalene and Suprascapular Blocks Used in Arthroscopic Shoulder Surgery
- Retrolaminar Block Versus Subcostal Transversus Abdominis Plane Block in Liver Resection Surgery (NA)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Bupivacaine hydrochloride 1% CI brief — competitive landscape report
- Bupivacaine hydrochloride 1% updates RSS · CI watch RSS
- Express Specialty Pharmacy portfolio CI
Frequently asked questions about Bupivacaine hydrochloride 1%
What is Bupivacaine hydrochloride 1%?
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Related
- Drug class: All Local anesthetic drugs
- Target: All drugs targeting Voltage-gated sodium channels
- Manufacturer: Express Specialty Pharmacy — full pipeline
- Therapeutic area: All drugs in Oncology
- Indication: Drugs for Local anesthesia
- Also known as: Bupivacaine hydrochloride
- Compare: Bupivacaine hydrochloride 1% vs similar drugs
- Pricing: Bupivacaine hydrochloride 1% cost, discount & access