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aprotinin or tranexamic acid

German Heart Center · Phase 3 active Small molecule

Tranexamic acid works by inhibiting the activation of plasminogen to plasmin, thereby reducing fibrinolysis and preventing excessive bleeding.

Tranexamic acid works by inhibiting the activation of plasminogen to plasmin, thereby reducing fibrinolysis and preventing excessive bleeding. Used for Surgical bleeding, Menorrhagia.

At a glance

Generic nameaprotinin or tranexamic acid
SponsorGerman Heart Center
Drug classAntifibrinolytic
ModalitySmall molecule
Therapeutic areaCardiovascular
PhasePhase 3

Mechanism of action

Tranexamic acid is a synthetic derivative of the amino acid lysine. It binds to plasminogen and prevents its activation to plasmin, which is the primary enzyme responsible for fibrinolysis. By inhibiting fibrinolysis, tranexamic acid reduces the breakdown of blood clots and prevents excessive bleeding.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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