H1 receptor antagonist

This page covers all H1 receptor antagonist drugs tracked by Drug Landscape: marketed products and active clinical-stage compounds, targeting H1 receptor, Histamine H1 receptor, H1-receptor.

Targets

H1 receptor · Histamine H1 receptor · H1-receptor · H1 histamine receptor

Marketed (3)

• Hidra1 · Farmoquimica S.A. · Allergy
  Hidra1 is an antihistamine that works by blocking the action of histamine in the body.
• H1 Antihistaminics · Erasmus Medical Center · Allergy/Immunology
  H1 antihistaminics block histamine H1 receptors on cell surfaces, preventing histamine-mediated allergic and inflammatory responses.
• olopatadine 0.2% ophthalmic solution · Allergan · Ophthalmology
  Olopatadine blocks H1-receptors on ocular mast cells and other immune cells to reduce histamine-mediated itching and allergic inflammation in the eye.

Phase 3 pipeline (2)

• Bepotastine besilate formulation · Bausch & Lomb Incorporated · Ophthalmology / Allergy
  Bepotastine besilate is a selective H1-receptor antagonist that blocks histamine signaling to reduce allergic symptoms.
• H1 Receptor Antagonist · Merck Sharp & Dohme LLC · Allergy/Immunology
  H1 receptor antagonists block histamine binding to H1 receptors, reducing histamine-mediated allergic and inflammatory responses.

Phase 2 pipeline (3)

• Bilastine 0.6% · Faes Farma, S.A. · Allergy
  Bilastine is an antihistamine that works by blocking the action of histamine, a substance in the body that causes allergy symptoms.
• H1 antihistamines · Genentech, Inc. · Respiratory
  Blocks H1 histamine receptors
• Bilastine 0.4% · Faes Farma, S.A. · Allergy
  Bilastine is an antihistamine that works by blocking the action of histamine, a substance in the body that causes allergy symptoms.