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Levocetirizine (drug) — Competitive Intelligence Brief
marketed
H1-receptor antagonist (second-generation antihistamine)
H1-receptor
Allergy/Immunology
Small molecule
Live · refreshed every 30 min
Target snapshot
Levocetirizine (drug) (Levocetirizine (drug)) — UCB Pharma. Levocetirizine is a selective H1-receptor antagonist that blocks histamine binding to H1 receptors on mast cells and basophils, preventing allergic cascade activation.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Levocetirizine (drug) TARGET | Levocetirizine (drug) | UCB Pharma | marketed | H1-receptor antagonist (second-generation antihistamine) | H1-receptor | |
| Bepreve | BEPOTASTINE | Bausch Health | marketed | Histamine-1 Receptor Antagonist | H1-receptor, mast cells | 2009-01-01 |
| bepotastine besilate ophthalmic solution | bepotastine besilate ophthalmic solution | Bausch & Lomb Incorporated | marketed | H1-receptor, mast cells | ||
| olopatadine 0.2% ophthalmic solution | olopatadine 0.2% ophthalmic solution | Allergan | marketed | H1-receptor antagonist | H1-receptor | |
| Cetirizine Dry Syrup | Cetirizine Dry Syrup | GlaxoSmithKline | phase 3 | H1-receptor antagonist (second-generation antihistamine) | H1-receptor | |
| Antihistamine Cetirizine Hydrochloride | Antihistamine Cetirizine Hydrochloride | Goldman, Butterwick, Fitzpatrick and Groff | marketed | H1-receptor antagonist (second-generation antihistamine) | H1 histamine receptor | |
| Cetirizine (Zyrtec) | Cetirizine (Zyrtec) | Organon and Co | marketed | H1-receptor antagonist (second-generation antihistamine) | H1 receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (H1-receptor antagonist (second-generation antihistamine) class)
- UCB Pharma · 5 drugs in this class
- Organon and Co · 3 drugs in this class
- Brian J Lipworth · 1 drug in this class
- GlaxoSmithKline · 1 drug in this class
- Goldman, Butterwick, Fitzpatrick and Groff · 1 drug in this class
- HK inno.N Corporation · 1 drug in this class
- AAADRS Clinical Research Center · 1 drug in this class
- University Hospital, Grenoble · 1 drug in this class
- Azienda Ospedaliera OO.RR. S. Giovanni di Dio e Ruggi D'Aragona · 1 drug in this class
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- Levocetirizine (drug) CI watch — RSS
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- Levocetirizine (drug) CI watch — JSON
- Levocetirizine (drug) alone — RSS
- Whole H1-receptor antagonist (second-generation antihistamine) class — RSS
Cite this brief
Drug Landscape (2026). Levocetirizine (drug) — Competitive Intelligence Brief. https://druglandscape.com/ci/levocetirizine-drug. Accessed 2026-05-16.
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