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Traditional anticoagulation

University of Sao Paulo General Hospital · FDA-approved active Small molecule Under review

Traditional anticoagulation is a Anticoagulant Small molecule drug developed by University of Sao Paulo General Hospital. It is currently FDA-approved for Atrial fibrillation for stroke prevention, Venous thromboembolism (DVT/PE) treatment and prophylaxis, Mechanical heart valve thromboprophylaxis. Also known as: Warfarin.

Traditional anticoagulation prevents blood clot formation by inhibiting coagulation cascade factors, typically through vitamin K antagonism or direct thrombin/factor Xa inhibition.

Traditional anticoagulation involves the use of medications such as rivaroxaban, which is an oligosaccharide modality, to prevent blood clot formation. It is studied in various conditions including peripheral arterial disease, stable and unstable angina, and is also used in combination with antithrombotic therapy.

At a glance

Generic nameTraditional anticoagulation
Also known asWarfarin
SponsorUniversity of Sao Paulo General Hospital
Drug classAnticoagulant
TargetVitamin K-dependent coagulation factors (II, VII, IX, X) or thrombin/Factor Xa
ModalitySmall molecule
Therapeutic areaCardiovascular
PhaseFDA-approved

Mechanism of action

Traditional anticoagulants work by interfering with the body's natural blood clotting cascade. Warfarin (a vitamin K antagonist) inhibits factors II, VII, IX, and X, while older parenteral agents like heparin inhibit thrombin and factor Xa directly. These mechanisms reduce the ability of blood to form pathological clots while maintaining hemostasis.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about Traditional anticoagulation

What is Traditional anticoagulation?

Traditional anticoagulation is a Anticoagulant drug developed by University of Sao Paulo General Hospital, indicated for Atrial fibrillation for stroke prevention, Venous thromboembolism (DVT/PE) treatment and prophylaxis, Mechanical heart valve thromboprophylaxis.

How does Traditional anticoagulation work?

Traditional anticoagulation prevents blood clot formation by inhibiting coagulation cascade factors, typically through vitamin K antagonism or direct thrombin/factor Xa inhibition.

What is Traditional anticoagulation used for?

Traditional anticoagulation is indicated for Atrial fibrillation for stroke prevention, Venous thromboembolism (DVT/PE) treatment and prophylaxis, Mechanical heart valve thromboprophylaxis, Acute coronary syndrome.

Who makes Traditional anticoagulation?

Traditional anticoagulation is developed and marketed by University of Sao Paulo General Hospital (see full University of Sao Paulo General Hospital pipeline at /company/university-of-sao-paulo-general-hospital).

Is Traditional anticoagulation also known as anything else?

Traditional anticoagulation is also known as Warfarin.

What drug class is Traditional anticoagulation in?

Traditional anticoagulation belongs to the Anticoagulant class. See all Anticoagulant drugs at /class/anticoagulant.

What development phase is Traditional anticoagulation in?

Traditional anticoagulation is FDA-approved (marketed).

What are the side effects of Traditional anticoagulation?

Common side effects of Traditional anticoagulation include Bleeding (major and minor), Bruising, Gastrointestinal bleeding, Intracranial hemorrhage, Warfarin necrosis (with warfarin).

What does Traditional anticoagulation target?

Traditional anticoagulation targets Vitamin K-dependent coagulation factors (II, VII, IX, X) or thrombin/Factor Xa and is a Anticoagulant.

Related

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing