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Remifentanil, propofol and citanest

University of Aarhus · FDA-approved active Small molecule

This is a combination of three anesthetic agents that work synergistically to induce and maintain general anesthesia through different mechanisms.

This is a combination of three anesthetic agents that work synergistically to induce and maintain general anesthesia through different mechanisms. Used for Induction and maintenance of general anesthesia for surgical procedures.

At a glance

Generic nameRemifentanil, propofol and citanest
SponsorUniversity of Aarhus
Drug classGeneral anesthetic combination
TargetMu opioid receptor (remifentanil); GABA-A receptor (propofol); Voltage-gated sodium channels (prilocaine)
ModalitySmall molecule
Therapeutic areaAnesthesiology
PhaseFDA-approved

Mechanism of action

Remifentanil is an opioid agonist that provides analgesia and sedation by binding to mu opioid receptors. Propofol is a sedative-hypnotic that enhances GABA-mediated inhibition in the central nervous system. Prilocaine (citanest) is a local anesthetic that blocks sodium channels in nerve membranes. Together, they provide rapid induction and maintenance of general anesthesia with analgesia.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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