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placebo and tramadol

University of Southern Denmark · FDA-approved active Small molecule Quality 2/100

Tramadol is a synthetic opioid analgesic that inhibits reuptake of norepinephrine and serotonin while also acting as a weak mu-opioid receptor agonist to provide pain relief.

Tramadol is a synthetic opioid analgesic that inhibits reuptake of norepinephrine and serotonin while also acting as a weak mu-opioid receptor agonist to provide pain relief. Used for Moderate pain management.

At a glance

Generic nameplacebo and tramadol
Also known asplacebo, Ultram
SponsorUniversity of Southern Denmark
Drug classOpioid analgesic with monoamine reuptake inhibition
TargetMu-opioid receptor; norepinephrine transporter; serotonin transporter
ModalitySmall molecule
Therapeutic areaPain Management
PhaseFDA-approved

Mechanism of action

Tramadol works through dual mechanisms: it binds to mu-opioid receptors in the central nervous system to produce analgesia, and it also inhibits the reuptake of norepinephrine and serotonin, enhancing their analgesic effects. This combination of opioid and monoamine reuptake inhibition makes it effective for moderate pain management. The placebo component in this study serves as a control comparator.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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