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LevoCept

Sebela Women's Health Inc. · Phase 3 active Small molecule

LevoCept is a selective estrogen receptor modulator (SERM) that modulates estrogen signaling to treat menopausal symptoms and related conditions in women.

LevoCept is a selective estrogen receptor modulator (SERM) that modulates estrogen signaling to treat menopausal symptoms and related conditions in women. Used for Vasomotor symptoms associated with menopause, Menopausal bone health and osteoporosis prevention.

At a glance

Generic nameLevoCept
Also known asLevonorgestrel-Releasing Intrauterine System
SponsorSebela Women's Health Inc.
Drug classSelective Estrogen Receptor Modulator (SERM)
TargetEstrogen receptor alpha (ERα) and estrogen receptor beta (ERβ)
ModalitySmall molecule
Therapeutic areaWomen's Health / Endocrinology
PhasePhase 3

Mechanism of action

LevoCept acts as a tissue-selective estrogen receptor modulator, binding to estrogen receptors with differential activity across tissues. This allows it to provide estrogen-like benefits in some tissues (such as bone and vasomotor symptom relief) while avoiding unwanted estrogenic effects in others (such as breast and endometrium), making it suitable for menopausal hormone therapy.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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