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LevoCept — Competitive Intelligence Brief
phase 3
Selective Estrogen Receptor Modulator (SERM)
Estrogen receptor alpha (ERα) and estrogen receptor beta (ERβ)
Women's Health / Endocrinology
Small molecule
Live · refreshed every 30 min
Target snapshot
LevoCept (LevoCept) — Sebela Women's Health Inc.. LevoCept is a selective estrogen receptor modulator (SERM) that modulates estrogen signaling to treat menopausal symptoms and related conditions in women.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| LevoCept TARGET | LevoCept | Sebela Women's Health Inc. | phase 3 | Selective Estrogen Receptor Modulator (SERM) | Estrogen receptor alpha (ERα) and estrogen receptor beta (ERβ) | |
| Bazedoxifene/Conjugated Estrogen | Bazedoxifene/Conjugated Estrogen | University of North Carolina, Chapel Hill | marketed | Selective Estrogen Receptor Modulator (SERM) combined with Conjugated Estrogens | Estrogen receptor alpha (ERα) and estrogen receptor beta (ERβ) | |
| Tamoxifen Oral Tablet | Tamoxifen Oral Tablet | Samsung Medical Center | marketed | Selective estrogen receptor modulator (SERM) | Estrogen receptor alpha (ERα) | |
| E2Nomac | E2Nomac | Sydney Centre for Reproductive Health Research | marketed | Selective Estrogen Receptor Modulator (SERM) | Estrogen receptor (ER-α/ER-β) | |
| fenofibrate and tibolone | fenofibrate and tibolone | Keogh Institute for Medical Research | marketed | Fibrate + Selective Estrogen Receptor Modulator (SERM) | PPAR-α (fenofibrate); Estrogen receptor, progesterone receptor, androgen receptor (tibolone) | |
| Metformin + Clomiphene | Metformin + Clomiphene | University of Auckland, New Zealand | marketed | Combination therapy: biguanide + selective estrogen receptor modulator (SERM) | Metformin: AMP-activated protein kinase (AMPK); Clomiphene: estrogen receptor (ER) | |
| tamoxifen citrate (Tamoxifen) | tamoxifen citrate (Tamoxifen) | H. Lee Moffitt Cancer Center and Research Institute | marketed | Selective estrogen receptor modulator (SERM) | Estrogen receptor alpha (ERα) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Selective Estrogen Receptor Modulator (SERM) class)
- Eli Lilly and Company · 1 drug in this class
- Sebela Women's Health Inc. · 1 drug in this class
- Sydney Centre for Reproductive Health Research · 1 drug in this class
- Wyeth is now a wholly owned subsidiary of Pfizer · 1 drug in this class
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Cite this brief
Drug Landscape (2026). LevoCept — Competitive Intelligence Brief. https://druglandscape.com/ci/levocept. Accessed 2026-05-13.
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