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Lantus, Amaryl

Sanofi · FDA-approved active Small molecule

Lantus, Amaryl is a Insulin analog (Lantus); Meglitinide/Sulfonylurea (Amaryl) Small molecule drug developed by Sanofi. It is currently FDA-approved for Type 2 diabetes mellitus, Type 1 diabetes mellitus (Lantus). Also known as: insulin glargine,glimepiride.

Lantus is a long-acting basal insulin that lowers blood glucose by promoting glucose uptake and utilization in peripheral tissues and inhibiting hepatic glucose production, while Amaryl is a meglitinide that stimulates pancreatic beta cells to release insulin in response to meals.

Lantus is a long-acting basal insulin that lowers blood glucose by promoting glucose uptake and utilization in peripheral tissues and inhibiting hepatic glucose production, while Amaryl is a meglitinide that stimulates pancreatic beta cells to release insulin in response to meals. Used for Type 2 diabetes mellitus, Type 1 diabetes mellitus (Lantus).

At a glance

Generic nameLantus, Amaryl
Also known asinsulin glargine,glimepiride
SponsorSanofi
Drug classInsulin analog (Lantus); Meglitinide/Sulfonylurea (Amaryl)
TargetInsulin receptor (Lantus); ATP-sensitive potassium channel on pancreatic beta cells (Amaryl)
ModalitySmall molecule
Therapeutic areaDiabetes
PhaseFDA-approved

Mechanism of action

Lantus (insulin glargine) is a recombinant human insulin analog with a prolonged duration of action (up to 24 hours), providing steady basal insulin coverage. Amaryl (glimepiride) is a short-acting insulin secretagogue that binds to ATP-sensitive potassium channels on beta cells, triggering insulin secretion primarily during and after meals. Together, they provide both basal and prandial insulin coverage for glycemic control.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about Lantus, Amaryl

What is Lantus, Amaryl?

Lantus, Amaryl is a Insulin analog (Lantus); Meglitinide/Sulfonylurea (Amaryl) drug developed by Sanofi, indicated for Type 2 diabetes mellitus, Type 1 diabetes mellitus (Lantus).

How does Lantus, Amaryl work?

Lantus is a long-acting basal insulin that lowers blood glucose by promoting glucose uptake and utilization in peripheral tissues and inhibiting hepatic glucose production, while Amaryl is a meglitinide that stimulates pancreatic beta cells to release insulin in response to meals.

What is Lantus, Amaryl used for?

Lantus, Amaryl is indicated for Type 2 diabetes mellitus, Type 1 diabetes mellitus (Lantus).

Who makes Lantus, Amaryl?

Lantus, Amaryl is developed and marketed by Sanofi (see full Sanofi pipeline at /company/sanofi).

Is Lantus, Amaryl also known as anything else?

Lantus, Amaryl is also known as insulin glargine,glimepiride.

What drug class is Lantus, Amaryl in?

Lantus, Amaryl belongs to the Insulin analog (Lantus); Meglitinide/Sulfonylurea (Amaryl) class. See all Insulin analog (Lantus); Meglitinide/Sulfonylurea (Amaryl) drugs at /class/insulin-analog-lantus-meglitinide-sulfonylurea-amaryl.

What development phase is Lantus, Amaryl in?

Lantus, Amaryl is FDA-approved (marketed).

What are the side effects of Lantus, Amaryl?

Common side effects of Lantus, Amaryl include Hypoglycemia, Weight gain, Injection site reactions (Lantus), Headache (Amaryl), Dizziness (Amaryl).

What does Lantus, Amaryl target?

Lantus, Amaryl targets Insulin receptor (Lantus); ATP-sensitive potassium channel on pancreatic beta cells (Amaryl) and is a Insulin analog (Lantus); Meglitinide/Sulfonylurea (Amaryl).

Related

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing