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Injection of Cyclosporin
Injection of Cyclosporin is a Calcineurin inhibitor Small molecule drug developed by Hospices Civils de Lyon. It is currently in Phase 3 development for Prevention of organ rejection in transplant recipients, Severe autoimmune conditions (e.g., severe rheumatoid arthritis, severe atopic dermatitis). Also known as: Cyclosporin A (CicloMulsion, verum).
Cyclosporin is a calcineurin inhibitor that suppresses T-cell activation by blocking the transcription of pro-inflammatory cytokines.
Cyclosporin is a calcineurin inhibitor that suppresses T-cell activation by blocking the transcription of pro-inflammatory cytokines. Used for Prevention of organ rejection in transplant recipients, Severe autoimmune conditions (e.g., severe rheumatoid arthritis, severe atopic dermatitis).
At a glance
| Generic name | Injection of Cyclosporin |
|---|---|
| Also known as | Cyclosporin A (CicloMulsion, verum) |
| Sponsor | Hospices Civils de Lyon |
| Drug class | Calcineurin inhibitor |
| Target | Calcineurin (protein phosphatase 2B) |
| Modality | Small molecule |
| Therapeutic area | Immunology |
| Phase | Phase 3 |
Mechanism of action
Cyclosporin binds to cyclophilin and inhibits calcineurin phosphatase, preventing dephosphorylation and nuclear translocation of NFAT (nuclear factor of activated T cells). This blocks the production of interleukin-2 and other cytokines essential for T-cell proliferation and immune response. The injectable formulation allows systemic immunosuppression for transplant rejection prevention and severe autoimmune conditions.
Approved indications
- Prevention of organ rejection in transplant recipients
- Severe autoimmune conditions (e.g., severe rheumatoid arthritis, severe atopic dermatitis)
Common side effects
- Nephrotoxicity
- Hypertension
- Tremor
- Gingival hyperplasia
- Hirsutism
- Infection
- Neurotoxicity (headache, paresthesia)
Key clinical trials
- Effects of Telitacicept vs Cyclophosphamide on Lupus Related Interstitial Lung Disease (PHASE4)
- Phase I Study of CTL Anti-DP Infusion Post-hematopoietic Stem Cell Transplantation (PHASE1)
- TRACK-TBI Precision Medicine Part 3 - Option II (PHASE2)
- Optimizing PTCy Dose and Timing (PHASE1, PHASE2)
- A Phase II Study of Zuberitamab Injection in Patients With Primary Membranous Nephropathy (PHASE2)
- A Phase Ib/ Ⅱ Clinical Study of MIL62 in Primary Membranous Nephropathy (PHASE1, PHASE2)
- Intralesional Cyclosporine for Alopecia Areata (EARLY_PHASE1)
- Cyclosporine and Prognosis in Acute Myocardial Infarction (MI) Patients (PHASE3)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Injection of Cyclosporin CI brief — competitive landscape report
- Injection of Cyclosporin updates RSS · CI watch RSS
- Hospices Civils de Lyon portfolio CI
Frequently asked questions about Injection of Cyclosporin
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Related
- Drug class: All Calcineurin inhibitor drugs
- Target: All drugs targeting Calcineurin (protein phosphatase 2B)
- Manufacturer: Hospices Civils de Lyon — full pipeline
- Therapeutic area: All drugs in Immunology
- Indication: Drugs for Prevention of organ rejection in transplant recipients
- Indication: Drugs for Severe autoimmune conditions (e.g., severe rheumatoid arthritis, severe atopic dermatitis)
- Also known as: Cyclosporin A (CicloMulsion, verum)
- Compare: Injection of Cyclosporin vs similar drugs
- Pricing: Injection of Cyclosporin cost, discount & access