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Duloxetine Hydrochloride (HCI)
Duloxetine Hydrochloride (HCI) is a Serotonin-norepinephrine reuptake inhibitor (SNRI) Small molecule drug developed by Eli Lilly and Company. It is currently in Phase 3 development for Major depressive disorder, Generalized anxiety disorder, Diabetic peripheral neuropathic pain. Also known as: LY248686, Cymbalta.
Duloxetine inhibits the reuptake of serotonin and norepinephrine in the central nervous system, increasing their availability at synaptic sites.
Duloxetine inhibits the reuptake of serotonin and norepinephrine in the central nervous system, increasing their availability at synaptic sites. Used for Major depressive disorder, Generalized anxiety disorder, Diabetic peripheral neuropathic pain.
At a glance
| Generic name | Duloxetine Hydrochloride (HCI) |
|---|---|
| Also known as | LY248686, Cymbalta |
| Sponsor | Eli Lilly and Company |
| Drug class | Serotonin-norepinephrine reuptake inhibitor (SNRI) |
| Target | Serotonin transporter (SERT); Norepinephrine transporter (NET) |
| Modality | Small molecule |
| Therapeutic area | Psychiatry, Neurology, Pain Management |
| Phase | Phase 3 |
Mechanism of action
Duloxetine is a serotonin-norepinephrine reuptake inhibitor (SNRI) that blocks the reuptake transporters for both serotonin and norepinephrine, leading to increased concentrations of these neurotransmitters in the synaptic cleft. This dual mechanism is thought to enhance mood regulation and pain signaling modulation. The drug is used to treat depression, anxiety disorders, and chronic pain conditions including diabetic peripheral neuropathic pain and fibromyalgia.
Approved indications
- Major depressive disorder
- Generalized anxiety disorder
- Diabetic peripheral neuropathic pain
- Fibromyalgia
- Chronic musculoskeletal pain
Common side effects
- Nausea
- Dizziness
- Somnolence
- Dry mouth
- Fatigue
- Constipation
- Decreased appetite
- Sweating
Key clinical trials
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Duloxetine Hydrochloride (HCI) CI brief — competitive landscape report
- Duloxetine Hydrochloride (HCI) updates RSS · CI watch RSS
- Eli Lilly and Company portfolio CI
Frequently asked questions about Duloxetine Hydrochloride (HCI)
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Related
- Drug class: All Serotonin-norepinephrine reuptake inhibitor (SNRI) drugs
- Target: All drugs targeting Serotonin transporter (SERT); Norepinephrine transporter (NET)
- Manufacturer: Eli Lilly and Company — full pipeline
- Therapeutic area: All drugs in Psychiatry, Neurology, Pain Management
- Indication: Drugs for Major depressive disorder
- Indication: Drugs for Generalized anxiety disorder
- Indication: Drugs for Diabetic peripheral neuropathic pain
- Also known as: LY248686, Cymbalta
- Compare: Duloxetine Hydrochloride (HCI) vs similar drugs
- Pricing: Duloxetine Hydrochloride (HCI) cost, discount & access