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Bifonazole spray twice daily

Bayer · Phase 2 active Small molecule

Bifonazole is an antifungal agent that works by inhibiting the synthesis of ergosterol, an essential component of fungal cell membranes.

Bifonazole is an antifungal agent that works by inhibiting the synthesis of ergosterol, an essential component of fungal cell membranes. Used for Cutaneous candidiasis, Dermatophytosis.

At a glance

Generic nameBifonazole spray twice daily
SponsorBayer
Drug classTriazole antifungal
TargetLanosterol 14α-demethylase
ModalitySmall molecule
Therapeutic areaDermatology
PhasePhase 2

Mechanism of action

Bifonazole is a triazole antifungal that binds to the fungal enzyme lanosterol 14α-demethylase, preventing the conversion of lanosterol to ergosterol. This disrupts the integrity of the fungal cell membrane, ultimately leading to cell death. Bifonazole is effective against a range of fungal pathogens, including dermatophytes and yeasts.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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