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Bifonazole spray once daily

Bayer · Phase 2 active Small molecule

Bifonazole is an antifungal agent that works by inhibiting the synthesis of ergosterol, an essential component of fungal cell membranes.

Bifonazole is an antifungal agent that works by inhibiting the synthesis of ergosterol, an essential component of fungal cell membranes. Used for Cutaneous candidiasis, Dermatophytosis.

At a glance

Generic nameBifonazole spray once daily
SponsorBayer
Drug classazole antifungal
Targetlanosterol 14α-demethylase
ModalitySmall molecule
Therapeutic areaInfectious Diseases
PhasePhase 2

Mechanism of action

Bifonazole achieves this by targeting the enzyme lanosterol 14α-demethylase, which is necessary for the conversion of lanosterol to ergosterol. This disruption of ergosterol synthesis ultimately leads to the death of fungal cells. Bifonazole is effective against a wide range of fungal pathogens, including dermatophytes, yeasts, and molds.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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