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Benzyl penicillin

KEMRI-Wellcome Trust Collaborative Research Program · Phase 3 active Small molecule ✓ Verified May 2026

Benzyl penicillin is a Beta-lactam antibiotic Small molecule drug developed by KEMRI-Wellcome Trust Collaborative Research Program. It is currently in Phase 3 development for Bacterial infections caused by susceptible organisms (gram-positive cocci, some gram-negative bacteria, and spirochetes), Pneumococcal infections, Streptococcal infections. Also known as: Medipen, Cristapen.

Benzyl penicillin inhibits bacterial cell wall synthesis by binding to penicillin-binding proteins and blocking peptidoglycan cross-linking.

Benzyl penicillin, also known as penicillin G, is a small molecule antibiotic used to treat various bacterial infections. It is indicated for conditions such as pneumonia, strep throat, syphilis, and others, but not typically for pneumococcal meningitis.

Likelihood of approval
60.3% vs 58.3% industry baseline
If approved by FDA: likely 2028–2030
Steps remaining: NDA/BLA submission
Confidence: High
Why this estimate
  • Baseline phase 3 → approval rate +58.3pp
    Industry-wide phase 3 drugs reach approval ~58.3% of the time (BIO/Informa 2023 industry benchmark across all therapeutic areas).
  • Anti-infectives pathway favourability +2.0pp
    Microbiological endpoints + non-inferiority designs raise approval rates above baseline.
Predicted approval windows by jurisdiction (conditional on FDA approval)
Regulator Country Likely year Lag vs FDA
FDA US 2028–2030
EMA EU 2029–2031 +0.7 yr
MHRA GB 2029–2031 +0.7 yr
Health Canada CA 2029–2032 +0.9 yr
TGA AU 2029–2032 +1.2 yr
PMDA JP 2029–2032 +1.5 yr
NMPA CN 2030–2033 +2.3 yr
MFDS KR 2029–2032 +1.4 yr
CDSCO IN 2029–2033 +1.8 yr
ANVISA BR 2030–2033 +2.3 yr

Hover any row for the lag rationale. Lag estimates are reduced when the drug has FDA Breakthrough or EMA PRIME designation (sponsors file globally in parallel).

Estimate based on the BIO/Informa industry phase transition rates plus per-drug modifiers for therapeutic area, sponsor type, FDA designations, mechanism, and trial design. Per-jurisdiction lags from Tufts CSDD international approval studies. Not investment, clinical or regulatory advice. Methodology: /methodology#likelihood.

At a glance

Generic nameBenzyl penicillin
Also known asMedipen, Cristapen
SponsorKEMRI-Wellcome Trust Collaborative Research Program
Drug classBeta-lactam antibiotic
TargetPenicillin-binding proteins (PBPs)
ModalitySmall molecule
Therapeutic areaInfectious Disease
PhasePhase 3

Mechanism of action

Benzyl penicillin (penicillin G) is a beta-lactam antibiotic that covalently binds to penicillin-binding proteins in susceptible bacteria, preventing the cross-linking of peptidoglycan strands in the cell wall. This disruption of cell wall integrity leads to bacterial cell lysis and death. It is bactericidal and effective against a broad range of gram-positive and some gram-negative bacteria.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

Competitive intelligence

For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:

Frequently asked questions about Benzyl penicillin

What is Benzyl penicillin?

Benzyl penicillin is a Beta-lactam antibiotic drug developed by KEMRI-Wellcome Trust Collaborative Research Program, indicated for Bacterial infections caused by susceptible organisms (gram-positive cocci, some gram-negative bacteria, and spirochetes), Pneumococcal infections, Streptococcal infections.

How does Benzyl penicillin work?

Benzyl penicillin inhibits bacterial cell wall synthesis by binding to penicillin-binding proteins and blocking peptidoglycan cross-linking.

What is Benzyl penicillin used for?

Benzyl penicillin is indicated for Bacterial infections caused by susceptible organisms (gram-positive cocci, some gram-negative bacteria, and spirochetes), Pneumococcal infections, Streptococcal infections, Meningitis.

Who makes Benzyl penicillin?

Benzyl penicillin is developed by KEMRI-Wellcome Trust Collaborative Research Program (see full KEMRI-Wellcome Trust Collaborative Research Program pipeline at /company/kemri-wellcome-trust-collaborative-research-program).

Is Benzyl penicillin also known as anything else?

Benzyl penicillin is also known as Medipen, Cristapen.

What drug class is Benzyl penicillin in?

Benzyl penicillin belongs to the Beta-lactam antibiotic class. See all Beta-lactam antibiotic drugs at /class/beta-lactam-antibiotic.

What development phase is Benzyl penicillin in?

Benzyl penicillin is in Phase 3.

What are the side effects of Benzyl penicillin?

Common side effects of Benzyl penicillin include Hypersensitivity reactions (rash, urticaria), Anaphylaxis, Diarrhea, Nausea, Seizures (high doses, renal impairment).

What does Benzyl penicillin target?

Benzyl penicillin targets Penicillin-binding proteins (PBPs) and is a Beta-lactam antibiotic.

Related

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing