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BCI-540

BrainCells Inc. · Phase 2 active Small molecule

BCI-540 is a small molecule that modulates the activity of GABA_A receptors.

BCI-540 is a small molecule that modulates the activity of GABA_A receptors. Used for Major depressive disorder, Generalized anxiety disorder.

At a glance

Generic nameBCI-540
SponsorBrainCells Inc.
Drug classGABA_A receptor modulator
TargetGABA_A receptor
ModalitySmall molecule
Therapeutic areaNeurology
PhasePhase 2

Mechanism of action

BCI-540 acts as a positive allosteric modulator of GABA_A receptors, enhancing the inhibitory effects of GABA. This mechanism is thought to contribute to its potential therapeutic effects in various neurological disorders.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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