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acamprosate (Campral)

University of North Carolina, Chapel Hill · FDA-approved active Small molecule

acamprosate (Campral) is a NMDA receptor modulator Small molecule drug developed by University of North Carolina, Chapel Hill. It is currently FDA-approved for Maintenance of abstinence in alcohol-dependent patients. Also known as: Acamprosate(Campral), Acamprosate, campral, alcohol dependence medication.

Acamprosate modulates glutamate and GABA neurotransmission to restore neurochemical balance disrupted by chronic alcohol use.

Acamprosate modulates glutamate and GABA neurotransmission to restore neurochemical balance disrupted by chronic alcohol use. Used for Maintenance of abstinence in alcohol-dependent patients.

At a glance

Generic nameacamprosate (Campral)
Also known asAcamprosate(Campral), Acamprosate, campral, alcohol dependence medication
SponsorUniversity of North Carolina, Chapel Hill
Drug classNMDA receptor modulator
TargetNMDA receptor (glutamate); GABA system
ModalitySmall molecule
Therapeutic areaPsychiatry / Addiction Medicine
PhaseFDA-approved

Mechanism of action

Acamprosate is believed to act as a weak antagonist at NMDA receptors and may enhance GABA-mediated inhibitory neurotransmission, helping to normalize the hyperexcitable state of the central nervous system that develops during alcohol dependence. By restoring glutamate-GABA balance, it reduces cravings and protects against relapse in alcohol-dependent patients who have achieved abstinence.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

Competitive intelligence

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Frequently asked questions about acamprosate (Campral)

What is acamprosate (Campral)?

acamprosate (Campral) is a NMDA receptor modulator drug developed by University of North Carolina, Chapel Hill, indicated for Maintenance of abstinence in alcohol-dependent patients.

How does acamprosate (Campral) work?

Acamprosate modulates glutamate and GABA neurotransmission to restore neurochemical balance disrupted by chronic alcohol use.

What is acamprosate (Campral) used for?

acamprosate (Campral) is indicated for Maintenance of abstinence in alcohol-dependent patients.

Who makes acamprosate (Campral)?

acamprosate (Campral) is developed and marketed by University of North Carolina, Chapel Hill (see full University of North Carolina, Chapel Hill pipeline at /company/university-of-north-carolina-chapel-hill).

Is acamprosate (Campral) also known as anything else?

acamprosate (Campral) is also known as Acamprosate(Campral), Acamprosate, campral, alcohol dependence medication.

What drug class is acamprosate (Campral) in?

acamprosate (Campral) belongs to the NMDA receptor modulator class. See all NMDA receptor modulator drugs at /class/nmda-receptor-modulator.

What development phase is acamprosate (Campral) in?

acamprosate (Campral) is FDA-approved (marketed).

What are the side effects of acamprosate (Campral)?

Common side effects of acamprosate (Campral) include Diarrhea, Headache, Nausea, Asthenia/weakness, Anxiety.

What does acamprosate (Campral) target?

acamprosate (Campral) targets NMDA receptor (glutamate); GABA system and is a NMDA receptor modulator.

Related

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing