Local anesthetic with adjuvant alpha-2 agonist
This page covers all Local anesthetic with adjuvant alpha-2 agonist drugs tracked by Drug Landscape: marketed products and active clinical-stage compounds, targeting Voltage-gated sodium channels (ropivacaine); alpha-2 adrenergic receptors (clonidine), Alpha-2 adrenergic receptor (clonidine); voltage-gated sodium channels (levobupivacaine).
Targets
Voltage-gated sodium channels (ropivacaine); alpha-2 adrenergic receptors (clonidine) · Alpha-2 adrenergic receptor (clonidine); voltage-gated sodium channels (levobupivacaine)
Marketed (2)
- ropivacaine plus clonidine · University Hospital, Lille · Anesthesia
Ropivacaine blocks sodium channels to provide local anesthesia, while clonidine enhances analgesia by activating alpha-2 adrenergic receptors. - clonidine, levobupivacaine · University Hospital Dubrava · Anesthesia and Pain Management
Clonidine is an alpha-2 adrenergic agonist that reduces pain signaling, while levobupivacaine is a local anesthetic that blocks sodium channels to prevent nerve conduction.
Patent intelligence
- local anesthetic with adjuvant alpha 2 agonist patent landscape — aggregated cliff calendar, attackable patents, originator estates