GABA receptor agonist

This page covers all GABA receptor agonist drugs tracked by Drug Landscape: marketed products and active clinical-stage compounds, targeting GABA_A receptor, alpha2-delta subunit of voltage-gated calcium channels, GABA_B receptor.

Targets

GABA_A receptor · alpha2-delta subunit of voltage-gated calcium channels · GABA_B receptor

Phase 3 pipeline (3)

• Propofol-Lipuro · University Hospital, Grenoble · Anesthesiology
  Propofol-Lipuro is a short-acting sedative-hypnotic agent that induces and maintains anesthesia by enhancing inhibitory neurotransmission mediated by GABA.
• propofol (drug) · B. Braun Melsungen AG · Anesthesiology
  Propofol is a short-acting sedative-hypnotic agent that acts on the central nervous system to induce and maintain anesthesia.
• placebo and pregabalin · Pfizer's Upjohn has merged with Mylan to form Viatris Inc. · Pain, Anxiety
  Pregabalin is a structural analog of the neurotransmitter gamma-aminobutyric acid (GABA) and acts as a GABA receptor agonist.

Phase 2 pipeline (2)

• Intrathecal Baclofen Pump · Amsterdam UMC, location VUmc · Neurology
  GABA_B receptor agonist
• Baclofen IR · Impax Laboratories, LLC · Neurology
  Baclofen IR is a central nervous system depressant that acts as a GABA_B receptor agonist.