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Regadenoson MRI myocardial blood flow — Competitive Intelligence Brief

Regadenoson MRI myocardial blood flow (Regadenoson MRI myocardial blood flow) competitive landscape: 6 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: Adenosine A2A receptor agonist. Area: Cardiovascular.

marketed Adenosine A2A receptor agonist Adenosine A2A receptor Cardiovascular Small molecule Live · refreshed every 30 min

Target snapshot

Regadenoson MRI myocardial blood flow (Regadenoson MRI myocardial blood flow) — University of Colorado, Denver. Regadenoson is a selective adenosine A2A receptor agonist that increases coronary blood flow to enable assessment of myocardial perfusion during cardiac MRI imaging.

Comparator set (6 drugs)

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
Regadenoson MRI myocardial blood flow TARGET Regadenoson MRI myocardial blood flow University of Colorado, Denver marketed Adenosine A2A receptor agonist Adenosine A2A receptor
Regadenoson myocardial perfusion imaging Regadenoson myocardial perfusion imaging University of Colorado, Denver marketed Adenosine A2A receptor agonist Adenosine A2A receptor
Regadenoson (Lexiscan) Regadenoson (Lexiscan) Brigham and Women's Hospital marketed Adenosine A2A receptor agonist Adenosine A2A receptor
Regadenoson peripheral - peripheral Regadenoson peripheral - peripheral Lokien van Nunen phase 3 Adenosine A2A receptor agonist Adenosine A2A receptor
Istradefylline (KW-6002) Istradefylline (KW-6002) Kyowa Kirin, Inc. phase 3 Adenosine A2A receptor antagonist Adenosine A2A receptor
AD109 AD109 Apnimed phase 3 Adenosine A2A receptor antagonist Adenosine A2A receptor
Pharmacological stress agents Pharmacological stress agents GE Healthcare phase 3 Cardiac stress agents Adenosine A2A receptor (adenosine); dopamine and beta-adrenergic receptors (dobutamine); adenosine A2A receptor (regadenoson)

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (Adenosine A2A receptor agonist class)

  1. Lokien van Nunen · 2 drugs in this class
  2. University of Colorado, Denver · 2 drugs in this class
  3. Brigham and Women's Hospital · 1 drug in this class

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Cite this brief

Drug Landscape (2026). Regadenoson MRI myocardial blood flow — Competitive Intelligence Brief. https://druglandscape.com/ci/regadenoson-mri-myocardial-blood-flow. Accessed 2026-05-17.

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