Last reviewed · How we verify
Metformin continue — Competitive Intelligence Brief
marketed
Biguanide
AMP-activated protein kinase (AMPK); mitochondrial complex I
Endocrinology/Diabetes
Small molecule
Live · refreshed every 30 min
Target snapshot
Metformin continue (Metformin continue) — University of Texas Southwestern Medical Center. Metformin reduces hepatic glucose production and improves insulin sensitivity, thereby lowering blood glucose levels in type 2 diabetes.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Metformin continue TARGET | Metformin continue | University of Texas Southwestern Medical Center | marketed | Biguanide | AMP-activated protein kinase (AMPK); mitochondrial complex I | |
| Placebo plus metformin | Placebo plus metformin | University Magna Graecia | marketed | Biguanide | AMP-activated protein kinase (AMPK), mitochondrial glycerophosphate dehydrogenase | |
| Metformin / Placebo treatment for 4 months | Metformin / Placebo treatment for 4 months | Norwegian University of Science and Technology | marketed | Biguanide | AMP-activated protein kinase (AMPK); mitochondrial glycerophosphate dehydrogenase | |
| Metformin + Clomiphene | Metformin + Clomiphene | University of Auckland, New Zealand | marketed | Combination therapy: biguanide + selective estrogen receptor modulator (SERM) | Metformin: AMP-activated protein kinase (AMPK); Clomiphene: estrogen receptor (ER) | |
| metformin+ gliclazide | metformin+ gliclazide | GlaxoSmithKline | marketed | Antidiabetic combination (biguanide + sulfonylurea) | Metformin: mitochondrial glycerophosphate dehydrogenase; Gliclazide: ATP-sensitive potassium channels on pancreatic beta cells | |
| Linagliptin / Metformin Oral Tablet | Linagliptin / Metformin Oral Tablet | Universidad de Guanajuato | marketed | DPP-4 inhibitor / Biguanide combination | DPP-4 (dipeptidyl peptidase-4) / AMPK pathway | |
| medical nutrition therapy + metformin | medical nutrition therapy + metformin | Instituto Nacional de Perinatologia Isidro Espinosa de los Reyes | marketed | Combination therapy: dietary intervention + biguanide antidiabetic | AMP-activated protein kinase (AMPK) and hepatic glucose metabolism (metformin component) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Biguanide class)
- AstraZeneca · 4 drugs in this class
- Merck Sharp & Dohme LLC · 3 drugs in this class
- University of Texas Southwestern Medical Center · 2 drugs in this class
- Mount Sinai Hospital, Canada · 2 drugs in this class
- GlaxoSmithKline · 2 drugs in this class
- Eli Lilly and Company · 2 drugs in this class
- University Magna Graecia · 2 drugs in this class
- First Affiliated Hospital of Wenzhou Medical University · 1 drug in this class
- Ente Ospedaliero Ospedali Galliera · 1 drug in this class
- Daewoong Pharmaceutical Co. LTD. · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Metformin continue — Competitive Intelligence Brief. https://druglandscape.com/ci/metformin-continue. Accessed 2026-05-13.
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