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Iniparib (SAR240550/BSI-201) — Competitive Intelligence Brief

Iniparib (SAR240550/BSI-201) (Iniparib (SAR240550/BSI-201)) competitive landscape: 6 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: PARP inhibitor. Area: Oncology.

phase 3 PARP inhibitor PARP (poly(ADP-ribose) polymerase) Oncology Small molecule Live · refreshed every 30 min

Target snapshot

Iniparib (SAR240550/BSI-201) (Iniparib (SAR240550/BSI-201)) — Sanofi. Iniparib inhibits poly(ADP-ribose) polymerase (PARP), an enzyme involved in DNA repair, thereby sensitizing cancer cells to chemotherapy and radiation.

Comparator set (6 drugs)

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
Iniparib (SAR240550/BSI-201) TARGET Iniparib (SAR240550/BSI-201) Sanofi phase 3 PARP inhibitor PARP (poly(ADP-ribose) polymerase)
Talazoparib with enzalutamide talazoparib-with-enzalutamide Pfizer marketed PARP inhibitor and androgen receptor inhibitor PARP enzymes and androgen receptor Not yet launched
Pharmacokinetics, Dosage of Niraparib Pharmacokinetics, Dosage of Niraparib Hospices Civils de Lyon marketed PARP inhibitor PARP1, PARP2
Olaparib Treatment D Olaparib Treatment D AstraZeneca marketed PARP inhibitor PARP1, PARP2
Talzenna Talazoparib Tosylate Pfizer Inc. marketed PARP inhibitor PARP1 and PARP2 enzymes
Fuzuloparib , Abiraterone acetate and Prednisone Fuzuloparib , Abiraterone acetate and Prednisone Jiangsu HengRui Medicine Co., Ltd. phase 3 PARP inhibitor (fuzuloparib) combined with CYP17A1 inhibitor (abiraterone acetate) and glucocorticoid (prednisone) PARP1/PARP2 (fuzuloparib); CYP17A1 (abiraterone acetate); glucocorticoid receptor (prednisone)
Saruparib (AZD5305) Saruparib (AZD5305) AstraZeneca phase 3 PARP inhibitor PARP1, PARP2

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (PARP inhibitor class)

  1. AstraZeneca · 5 drugs in this class
  2. BeiGene · 2 drugs in this class
  3. Clovis Oncology, Inc. · 1 drug in this class
  4. Fondazione Ricerca Traslazionale · 1 drug in this class
  5. GERCOR - Multidisciplinary Oncology Cooperative Group · 1 drug in this class
  6. Hospices Civils de Lyon · 1 drug in this class
  7. Pfizer Inc. · 1 drug in this class
  8. Sanofi · 1 drug in this class
  9. Tesaro, Inc. · 1 drug in this class
  10. The First Affiliated Hospital of Xiamen University · 1 drug in this class

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Cite this brief

Drug Landscape (2026). Iniparib (SAR240550/BSI-201) — Competitive Intelligence Brief. https://druglandscape.com/ci/iniparib-sar240550-bsi-201. Accessed 2026-05-16.

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