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Inhaled Long-Acting Muscarinic Antagonist — Competitive Intelligence Brief
phase 3
Long-acting muscarinic antagonist (LAMA)
M3 muscarinic acetylcholine receptor
Respiratory / Pulmonology
Small molecule
Live · refreshed every 30 min
Target snapshot
Inhaled Long-Acting Muscarinic Antagonist (Inhaled Long-Acting Muscarinic Antagonist) — Sanofi. Blocks muscarinic acetylcholine receptors in the airways to reduce bronchoconstriction and mucus secretion in chronic respiratory diseases.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Inhaled Long-Acting Muscarinic Antagonist TARGET | Inhaled Long-Acting Muscarinic Antagonist | Sanofi | phase 3 | Long-acting muscarinic antagonist (LAMA) | M3 muscarinic acetylcholine receptor | |
| Drug: ipratropium (AtroventTM) | Drug: ipratropium (AtroventTM) | AstraZeneca | marketed | Anticholinergic bronchodilator | M3 muscarinic acetylcholine receptor | |
| Albuterol, ipratropium bromide | Albuterol, ipratropium bromide | Children's Hospital of Philadelphia | marketed | Combination bronchodilator (beta-2 agonist + anticholinergic) | Beta-2 adrenergic receptor; M3 muscarinic acetylcholine receptor | |
| solifenacin succinate suspension | solifenacin succinate suspension | Astellas Pharma Inc | marketed | Muscarinic M3 receptor antagonist | M3 muscarinic acetylcholine receptor | |
| Toviaz (Fesoterodine) | Toviaz (Fesoterodine) | Weill Medical College of Cornell University | marketed | Muscarinic M3 receptor antagonist | M3 muscarinic acetylcholine receptor | |
| salbutamol + ipratropium bromide nebules | salbutamol + ipratropium bromide nebules | Imperial College London | marketed | Combination bronchodilator (beta-2 agonist + anticholinergic) | Beta-2 adrenergic receptor (salbutamol); M3 muscarinic acetylcholine receptor (ipratropium) | |
| Solifenacin for 24 weeks | Solifenacin for 24 weeks | National Taiwan University Hospital | marketed | Muscarinic M3 receptor antagonist | M3 muscarinic acetylcholine receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Long-acting muscarinic antagonist (LAMA) class)
- GlaxoSmithKline · 9 drugs in this class
- AstraZeneca · 3 drugs in this class
- Chia Tai Tianqing Pharmaceutical Group Co., Ltd. · 1 drug in this class
- Chiesi Farmaceutici S.p.A. · 1 drug in this class
- IRCCS Azienda Ospedaliero-Universitaria di Bologna · 1 drug in this class
- Lupin, Inc. · 1 drug in this class
- Sanofi · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Inhaled Long-Acting Muscarinic Antagonist — Competitive Intelligence Brief. https://druglandscape.com/ci/inhaled-long-acting-muscarinic-antagonist. Accessed 2026-05-17.
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