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Estriol Cream 0.1% — Competitive Intelligence Brief
marketed
Estrogen receptor agonist
Estrogen receptor alpha (ERα) and estrogen receptor beta (ERβ)
Gynecology / Menopause
Small molecule
Live · refreshed every 30 min
Target snapshot
Estriol Cream 0.1% (Estriol Cream 0.1%) — Dr. August Wolff GmbH & Co. KG Arzneimittel. Estriol is a weak estrogen that binds to estrogen receptors in vaginal and urogenital tissues to restore epithelial maturation and improve local tissue health.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Estriol Cream 0.1% TARGET | Estriol Cream 0.1% | Dr. August Wolff GmbH & Co. KG Arzneimittel | marketed | Estrogen receptor agonist | Estrogen receptor alpha (ERα) and estrogen receptor beta (ERβ) | |
| estriol cream | estriol cream | Hatice Tukenmez Kurnaz | marketed | Estrogen receptor agonist | Estrogen receptor alpha (ERα) and estrogen receptor beta (ERβ) | |
| Vaginal estradiol tablets | Vaginal estradiol tablets | Johns Hopkins University | marketed | Estrogen receptor agonist | Estrogen receptor alpha (ERα) and estrogen receptor beta (ERβ) | |
| estradiol valerat | estradiol valerat | farzaneh hojjat | marketed | Estrogen receptor agonist | Estrogen receptor alpha (ERα), Estrogen receptor beta (ERβ) | |
| Estradiol 0.01% Vag Cream | Estradiol 0.01% Vag Cream | TriHealth Inc. | marketed | Estrogen receptor agonist | Estrogen receptor alpha (ERα) and estrogen receptor beta (ERβ) | |
| Estradiol (E2) | Estradiol (E2) | Martin Blomberg Jensen | phase 3 | Estrogen receptor agonist | Estrogen receptor alpha (ERα), Estrogen receptor beta (ERβ) | |
| Generic Estradiol Vaginal Cream USP, 0.01% | Generic Estradiol Vaginal Cream USP, 0.01% | Actavis Inc. | phase 3 | Estrogen receptor agonist | Estrogen receptor alpha (ERα), Estrogen receptor beta (ERβ) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Estrogen receptor agonist class)
- Actavis Inc. · 1 drug in this class
- Bayer · 1 drug in this class
- Dr. August Wolff GmbH & Co. KG Arzneimittel · 1 drug in this class
- Hatice Tukenmez Kurnaz · 1 drug in this class
- Johns Hopkins University · 1 drug in this class
- Martin Blomberg Jensen · 1 drug in this class
- TriHealth Inc. · 1 drug in this class
- farzaneh hojjat · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Estriol Cream 0.1% — Competitive Intelligence Brief. https://druglandscape.com/ci/estriol-cream-0-1. Accessed 2026-05-16.
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