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Mektovi — Competitive Intelligence Brief
discontinued
Dual specificity mitogen-activated protein kinase kinase 1
Oncology
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Target snapshot
Mektovi (binimetinib) — Pfizer. Mektovi works by blocking a specific enzyme called MEK1, which is involved in sending signals that promote cancer cell growth.
Comparator set (2 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Mektovi TARGET | binimetinib | Pfizer | discontinued | Dual specificity mitogen-activated protein kinase kinase 1 | 2018-01-01 | |
| Mektovi | mek162 | Pfizer | marketed | Dual specificity mitogen-activated protein kinase kinase 1 | 2018-01-01 | |
| Cotellic | cobimetinib | Roche | marketed | Kinase Inhibitor | Dual specificity mitogen-activated protein kinase kinase 1 | 2015-01-01 |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
- — Mektovi · 9850229 · US
- — Mektovi · 10005761 · US
- — Mektovi · 9314464 · US
- — Mektovi · 9562016 · US
- — Mektovi · 9598376 · US
- — Mektovi · 9980944 · US
Sponsor landscape
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Cite this brief
Drug Landscape (2026). Mektovi — Competitive Intelligence Brief. https://druglandscape.com/ci/binimetinib. Accessed 2026-05-13.
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