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Mektovi — Competitive Intelligence Brief

Mektovi (binimetinib) competitive landscape: 2 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Area: Oncology.

discontinued Dual specificity mitogen-activated protein kinase kinase 1 Oncology Live · refreshed every 30 min

Target snapshot

Mektovi (binimetinib) — Pfizer. Mektovi works by blocking a specific enzyme called MEK1, which is involved in sending signals that promote cancer cell growth.

Comparator set (2 drugs)

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
Mektovi TARGET binimetinib Pfizer discontinued Dual specificity mitogen-activated protein kinase kinase 1 2018-01-01
Mektovi mek162 Pfizer marketed Dual specificity mitogen-activated protein kinase kinase 1 2018-01-01
Cotellic cobimetinib Roche marketed Kinase Inhibitor Dual specificity mitogen-activated protein kinase kinase 1 2015-01-01

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

Sponsor landscape

No sponsor landscape data.

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Cite this brief

Drug Landscape (2026). Mektovi — Competitive Intelligence Brief. https://druglandscape.com/ci/binimetinib. Accessed 2026-05-13.

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