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Abiraterone acetate, Prednisolone — Competitive Intelligence Brief
phase 2
CYP17A1 inhibitor (androgen synthesis inhibitor)
CYP17A1 (17α-hydroxylase/17,20-lyase)
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
Abiraterone acetate, Prednisolone (Abiraterone acetate, Prednisolone) — Cancer Trials Ireland. Abiraterone acetate inhibits CYP17A1 to block androgen synthesis, while prednisolone suppresses adrenocorticotropic hormone feedback to further reduce testosterone production in castration-resistant prostate cancer.
Comparator set (2 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Abiraterone acetate, Prednisolone TARGET | Abiraterone acetate, Prednisolone | Cancer Trials Ireland | phase 2 | CYP17A1 inhibitor (androgen synthesis inhibitor) | CYP17A1 (17α-hydroxylase/17,20-lyase) | |
| Abiraterone acetate and prednisone | Abiraterone acetate and prednisone | Janssen Research & Development, LLC | phase 3 | CYP17A1 inhibitor (androgen synthesis inhibitor) | CYP17A1 (17α-hydroxylase/17,20-lyase) | |
| Abiraterone + Prednisolone/Prednisone | Abiraterone + Prednisolone/Prednisone | AstraZeneca | phase 3 | CYP17A1 inhibitor (androgen synthesis inhibitor) + glucocorticoid | CYP17A1 (17α-hydroxylase/17,20-lyase) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (CYP17A1 inhibitor (androgen synthesis inhibitor) class)
- Cancer Trials Ireland · 1 drug in this class
- Janssen Research & Development, LLC · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Abiraterone acetate, Prednisolone — Competitive Intelligence Brief. https://druglandscape.com/ci/abiraterone-acetate-prednisolone. Accessed 2026-05-16.
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