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Abiraterone acetate MTD — Competitive Intelligence Brief
phase 1
CYP17 inhibitor
CYP17
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
Abiraterone acetate MTD (Abiraterone acetate MTD) — Cougar Biotechnology, Inc.. Androgen receptor inhibitor
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Abiraterone acetate MTD TARGET | Abiraterone acetate MTD | Cougar Biotechnology, Inc. | phase 1 | CYP17 inhibitor | CYP17 | |
| NIRAPARIB | NIRAPARIB | marketed | PARP-1, PARP-2, CYP17 | 2017-01-01 | ||
| Abiraterone Acetate | abiraterone | Pfizer | marketed | Androgen biosynthesis inhibitor | CYP17 | 2011-01-01 |
| Abiraterone + Prednisolone/Prednisone | Abiraterone + Prednisolone/Prednisone | AstraZeneca | phase 3 | CYP17A1 inhibitor (androgen synthesis inhibitor) + glucocorticoid | CYP17A1 (17α-hydroxylase/17,20-lyase) | |
| Abiraterone with Prednisone or Enzalutamide | Abiraterone with Prednisone or Enzalutamide | Curium US LLC | phase 3 | CYP17A1 inhibitor (abiraterone) + androgen receptor antagonist (enzalutamide) + glucocorticoid (prednisone) | CYP17A1 (abiraterone); androgen receptor (enzalutamide); glucocorticoid receptor (prednisone) | |
| Enzalutamide, Abiraterone | Enzalutamide, Abiraterone | Veru Inc. | phase 3 | Androgen receptor antagonist + CYP17A1 inhibitor combination | Androgen receptor (AR) and CYP17A1 | |
| Fuzuloparib , Abiraterone acetate and Prednisone | Fuzuloparib , Abiraterone acetate and Prednisone | Jiangsu HengRui Medicine Co., Ltd. | phase 3 | PARP inhibitor (fuzuloparib) combined with CYP17A1 inhibitor (abiraterone acetate) and glucocorticoid (prednisone) | PARP1/PARP2 (fuzuloparib); CYP17A1 (abiraterone acetate); glucocorticoid receptor (prednisone) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (CYP17 inhibitor class)
- Cougar Biotechnology, Inc. · 2 drugs in this class
- Janssen Research & Development, LLC · 2 drugs in this class
- Assistance Publique - Hôpitaux de Paris · 1 drug in this class
- Chia Tai Tianqing Pharmaceutical Group Co., Ltd. · 1 drug in this class
- GU Research Network, LLC · 1 drug in this class
- Han Xu, M.D., Ph.D., FAPCR, Sponsor-Investigator, IRB Chair · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Abiraterone acetate MTD — Competitive Intelligence Brief. https://druglandscape.com/ci/abiraterone-acetate-mtd. Accessed 2026-05-16.
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