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Abiraterone Acetate — Competitive Intelligence Brief
marketed
Androgen biosynthesis inhibitor
CYP17
Oncology
Live · refreshed every 30 min
Target snapshot
Abiraterone Acetate (abiraterone) — Pfizer. Abiraterone is an androgen biosynthesis inhibitor that targets CYP17 to reduce androgen production in prostate cancer cells.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Abiraterone Acetate TARGET | abiraterone | Pfizer | marketed | Androgen biosynthesis inhibitor | CYP17 | 2011-01-01 |
| NIRAPARIB | NIRAPARIB | marketed | PARP-1, PARP-2, CYP17 | 2017-01-01 | ||
| Abiraterone acetate and prednisone | Abiraterone acetate and prednisone | Janssen Research & Development, LLC | phase 3 | CYP17A1 inhibitor (androgen synthesis inhibitor) | CYP17A1 (17α-hydroxylase/17,20-lyase) | |
| Abiraterone Acetate (AA) | Abiraterone Acetate (AA) | Janssen Research & Development, LLC | phase 3 | CYP17A1 inhibitor | CYP17A1 (17α-hydroxylase/17,20-lyase) | |
| Fuzuloparib , Abiraterone acetate and Prednisone | Fuzuloparib , Abiraterone acetate and Prednisone | Jiangsu HengRui Medicine Co., Ltd. | phase 3 | PARP inhibitor (fuzuloparib) combined with CYP17A1 inhibitor (abiraterone acetate) and glucocorticoid (prednisone) | PARP1/PARP2 (fuzuloparib); CYP17A1 (abiraterone acetate); glucocorticoid receptor (prednisone) | |
| Abiraterone Acetate or Enzalutamide | Abiraterone Acetate or Enzalutamide | National Cancer Institute, Naples | phase 3 | Androgen synthesis inhibitor (abiraterone) / Androgen receptor antagonist (enzalutamide) | CYP17A1 (abiraterone) / Androgen receptor (enzalutamide) | |
| Abiraterone + Prednisolone/Prednisone | Abiraterone + Prednisolone/Prednisone | AstraZeneca | phase 3 | CYP17A1 inhibitor (androgen synthesis inhibitor) + glucocorticoid | CYP17A1 (17α-hydroxylase/17,20-lyase) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Androgen biosynthesis inhibitor class)
- Pfizer · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Abiraterone Acetate — Competitive Intelligence Brief. https://druglandscape.com/ci/abiraterone. Accessed 2026-05-13.
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