Last reviewed · How we verify

NCT06041646

Tachyphylaxis, Tolerance, & Withdrawal Post Treatment With Igalmi for Agitation in Schizophrenia or Bipolar Disorder

Completed Phase 4 Results posted Last updated 2 January 2026
What this trial tests

Phase 4 trial testing Sublingual film containing Igalmi in Bipolar Disorder in 29 participants. Completed in 29 April 2024.

Timeline
2 October 2023
Primary endpoint
29 April 2024
29 April 2024

Quick facts

Lead sponsorBioXcel Therapeutics Inc
PhasePhase 4
StatusCompleted
Study typeINTERVENTIONAL
Allocationna
Designsingle group
Maskingnone
Primary purposetreatment
Enrollment29
Start date2 October 2023
Primary completion29 April 2024
Estimated completion29 April 2024
Sites2 locations across United States

Drugs / interventions tested

Conditions studied

Sponsor

BioXcel Therapeutics Inc — full company profile →

Who can join

Adults 18 to 65, any sex, with Bipolar Disorder or Schizophrenia. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Change From Baseline in the Positive and Negative Syndrome Scale- Excited Component (PEC) Total Score Primary · Baseline and 2 hours post-dose for all doses administered over 7 days.

The Positive and Negative Syndrome Scale-Excited Component (PEC) includes 5 items-poor impulse control, tension, hostility, uncooperativeness, and excitement-each of which is rated from 1 (minimum) to 7 (maximum); the sum of these 5 items, the PEC total score, ranges from 5 (absence of agitation) to 35 (extremely severe).

Dose 1
GroupValue95% CI
Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)-10.4± 2.94
Dose 2
GroupValue95% CI
Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)-10.0± 3.54
Dose 3
GroupValue95% CI
Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)-10.1± 3.60
Dose 4
GroupValue95% CI
Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)-9.8± 2.55
Dose 5
GroupValue95% CI
Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)-11.5± 4.51
Dose 6
GroupValue95% CI
Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)-8.7± 3.79
Dose 7
GroupValue95% CI
Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)-11.0± NA
Clinical Global Impression - Improvement (CGI-I) Primary · 2 hours post-dose for all doses administered over 7 days.

The Clinical Global Impression - Improvement (CGI-I) for agitation in response to treatment measures the current level of agitation relative to the level of agitation prior to administration of study intervention. The CGI-I scores range from 1 to 7 with a score of 1 indicating very much improved, and a score of 7 indicating very much worse.

Dose 1
GroupValue95% CI
Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)1.2± 0.50
Dose 2
GroupValue95% CI
Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)1.2± 0.39
Dose 3
GroupValue95% CI
Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)1.3± 0.47
Dose 4
GroupValue95% CI
Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)1.0± 0.00
Dose 5
GroupValue95% CI
Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)1.2± 0.41
Dose 6
GroupValue95% CI
Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)1.3± 0.58
Dose 7
GroupValue95% CI
Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)2.0± NA
Number of Participants With Adverse Events During the Follow-up Period Secondary · Day 8 through Day 10

Evaluation of withdrawal phenomenon based on the occurrence of adverse events such as tachycardia, systolic hypertension, nausea, or vomiting and the emergence of any new adverse events on ≥2 consecutive days of the 3-day off-treatment follow-up period.

GroupValue95% CI
Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)0

Adverse events — posted to ClinicalTrials.gov

Time frame: 10 days. Reporting threshold: 3%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

Active Treatment - 180 mcg of Igalmi (Dexmedetomidine)
Serious: 0/28 (0%)
Deaths: 0/28
Other adverse events (17 terms — click to expand)

ReactionSystemActive Treatment - 180 mcg…
HeadacheNervous system disorders
SomnolenceNervous system disorders
Dry mouthGastrointestinal disorders
HypotensionVascular disorders
DizzinessNervous system disorders
SyncopeNervous system disorders
DyspepsiaGastrointestinal disorders
Gastroesophageal reflux diseaseGastrointestinal disorders
Hypoesthesia oralGastrointestinal disorders
Orthostatic hypotensionVascular disorders
ContusionInjury, poisoning and procedural complications
Limb injuryInjury, poisoning and procedural complications
Skin abrasionInjury, poisoning and procedural complications
Tongue injuryInjury, poisoning and procedural complications
ArthralgiaMusculoskeletal and connective tissue disorders
Back painMusculoskeletal and connective tissue disorders
DysmenorrheaReproductive system and breast disorders

Data from ClinicalTrials.gov NCT06041646 adverse events section.

Sponsor's own description

This is an in-clinic, single arm, open-label study assessing tachyphylaxis, tolerance, and withdrawal following repeated doses of Igalmi in adult males and females with agitation associated with schizophrenia or bipolar disorder.

Publications & conference data

1 peer-reviewed publication reference this trial (live from Europe PMC):

  1. ACNP 63rd Annual Meeting: Poster Abstracts P1-P304
    · 2024

Verify or expand the search:

Other recruiting trials for Bipolar Disorder

Currently open trials in the same condition.

Other BioXcel Therapeutics Inc trials

Trials by the same sponsor.

Verify against primary sources

Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT06041646.

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing