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NCT03782987

A Study in Healthy Men to Test How Itraconazole Influences the Amount of BI 730357 in the Blood

Completed Phase 1 Results posted Last updated 12 July 2023
What this trial tests

Phase 1 trial testing BI 730357 in Healthy in 14 participants. Completed in 11 March 2019.

Timeline
10 January 2019
Primary endpoint
11 March 2019
11 March 2019

Quick facts

Lead sponsorBoehringer Ingelheim
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationnon randomized
Designcrossover
Maskingnone
Primary purposetreatment
Enrollment14
Start date10 January 2019
Primary completion11 March 2019
Estimated completion11 March 2019
Sites1 location across Germany

Drugs / interventions tested

Conditions studied

Sponsor

Boehringer Ingelheim — full company profile →

Who can join

Adults 18 to 50, male only, with Healthy. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Area Under the Concentration-time Curve of the BI 730357 in Plasma Over the Time Interval From 0 to the Last Quantifiable Data Point (AUC0-tz) Primary · Pharmacokinetic samples were taken within 3 hours (h) before administration of BI 730357 and at 0.5, 1, 1.5, 2, 2.5, 3, 3.5, 4, 5, 6, 8, 12, 24, 34, 47, 71, 119 and 167 h in both periods and additionally at 215 and 263 h only for period 2.

AUC0-tz, area under the concentration-time curve of the BI 730357 in plasma over the time interval from 0 to the last quantifiable data point is presented.

GroupValue95% CI
BI 730357 + Itraconazole (T)43239.08± NA
BI 730357 (R)6657.49± NA
Maximum Measured Concentration of the BI 730357 in Plasma (Cmax) Primary · Pharmacokinetic samples were taken within 3 hours (h) before administration of BI 730357 and at 0.5, 1, 1.5, 2, 2.5, 3, 3.5, 4, 5, 6, 8, 12, 24, 34, 47, 71, 119 and 167 h in both periods and additionally at 215 and 263 h only for period 2.

Cmax, maximum measured concentration of the BI 730357 in plasma is presented here.

GroupValue95% CI
BI 730357 + Itraconazole (T)311.01± NA
BI 730357 (R)186.36± NA
Area Under the Concentration-time Curve of the BI 730357 in Plasma Over the Time Interval From 0 Extrapolated to Infinity (AUC0-∞) Secondary · Pharmacokinetic samples were taken within 3 hours (h) before administration of BI 730357 and at 0.5, 1, 1.5, 2, 2.5, 3, 3.5, 4, 5, 6, 8, 12, 24, 34, 47, 71, 119 and 167 h in both periods and additionally at 215 and 263 h only for period 2.

AUC0-∞, area under the concentration-time curve of the BI 730357 in plasma over the time interval from 0 extrapolated to infinity is presented here.

GroupValue95% CI
BI 730357 + Itraconazole (T)64934.55± NA
BI 730357 (R)6971.67± NA

Adverse events — posted to ClinicalTrials.gov

Time frame: BI 730357: From first administration of BI 730357, up to 168 hours. Itraconazole: From first administration of itraconazole until second administration of BI 730357, up to 73 hours. BI 730357+ Itraconazole: From second administration of BI 730357 until 216 hours after the last administration of itraconazole, up to 18 days.. Reporting threshold: 5%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

BI 730357 (R)
Serious: 0/14 (0%)
Deaths: 0/14
Itraconazole
Serious: 0/14 (0%)
Deaths: 0/14
BI 730357 + Itraconazole (T)
Serious: 0/14 (0%)
Deaths: 0/14
Other adverse events (11 terms — click to expand)

ReactionSystemBI 730357 (R)ItraconazoleBI 730357 + Itraconazole (T)
HeadacheNervous system disorders
DiarrhoeaGastrointestinal disorders
RhinitisInfections and infestations
NauseaGastrointestinal disorders
Vessel puncture site painGeneral disorders
Seasonal allergyImmune system disorders
NasopharyngitisInfections and infestations
ArthralgiaMusculoskeletal and connective tissue disorders
Musculoskeletal painMusculoskeletal and connective tissue disorders
MyalgiaMusculoskeletal and connective tissue disorders
PresyncopeNervous system disorders

Data from ClinicalTrials.gov NCT03782987 adverse events section.

Sponsor's own description

The main objective of this trial is to investigate the relative bioavailability of BI 730357 in plasma when given as oral single dose together with multiple oral doses of itraconazole (Test, T) as compared to when given alone as oral single dose (Reference, R)

Publications & conference data

1 peer-reviewed publication reference this trial (live from Europe PMC):

  1. Assessing Drug-Drug Interaction and Food Effect for BCS Class 2 Compound BI 730357 (Retinoic Acid-Related Orphan Receptor Gamma Antagonist, Bevurogant) Using a Physiology-Based Pharmacokinetics Modeling (PBPK) Approach with Semi-Mechanistic Absorption.
    Kanacher T, Sjögren E, Korell J, Plan EL, et al · · 2025 · PMID 40142978 · DOI 10.3390/pharmaceutics17030314

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Other trials of BI 730357

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Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT03782987.

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing