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NCT02163499

Open-label Safety and Efficacy of Sodium Zirconium Cyclosilicate for up to 12 Months

Completed Phase 3 Results posted Last updated 27 June 2018
What this trial tests

Phase 3 trial testing Sodium Zirconium Cyclosilicate in Hyperkalemia in 751 participants. Completed in 30 November 2016.

Timeline
30 June 2014
Primary endpoint
30 November 2016
30 November 2016

Quick facts

Lead sponsorZS Pharma, Inc.
PhasePhase 3
StatusCompleted
Study typeINTERVENTIONAL
Allocationna
Designsingle group
Maskingnone
Primary purposesupportive care
Enrollment751
Start date30 June 2014
Primary completion30 November 2016
Estimated completion30 November 2016
Sites50 locations across South Africa, Netherlands, United Kingdom, Germany, Romania, Australia, United States

Drugs / interventions tested

Conditions studied

Sponsor

ZS Pharma, Inc. — full company profile →

Who can join

18 and older, any sex, with Hyperkalemia. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Proportion of Subjects With Mean S-K Between 3.5 and 5.5 mmol/L, Inclusive Months 3 to 12 Secondary · Study Days 85 to 365

Proportion of Subjects with mean S-K between 3.5 and 5.5 mmol/L during Extended Dosing Phase - ITT Population

GroupValue95% CI
Proportion0.9850.972 – 0.993
Mean S-K Levels Months 3 to 12, Months 6 to 9, and Months 9 to 12. Secondary · Study days 85 to 365

Mean S-K levels months 3 to 12(EP Days 85, 113, 141, 176, 211, 239, 267, 295, 330, 365 and EOS),months 6 to 9, and months 9 to 12.

Acute Phase Baseline
GroupValue95% CI
Mean S-K Levels Months 3 to 12,6 to 9, and 9 to 125.59± 0.425
Extended Dosing Days 85 to 365/End of Study
GroupValue95% CI
Mean S-K Levels Months 3 to 12,6 to 9, and 9 to 124.66± 0.379
Extended Dosing Days 211 to 267
GroupValue95% CI
Mean S-K Levels Months 3 to 12,6 to 9, and 9 to 124.68± 0.404
Extended Dosing Days 295 to 365
GroupValue95% CI
Mean S-K Levels Months 3 to 12,6 to 9, and 9 to 124.62± 0.401
Percent of Participants With Restoration of Normal Serum Potassium (S-K) Values (3.5 to 5.0 mmol/L, Inclusive) at the End of the Acute Phase Primary · 72 Hours

Percentage of subjects with S-K values between 3.5 and 5.0 mmol/L, inclusive at the end of the Acute Phase - ITT Population

GroupValue95% CI
Percentage77.974.8 – 80.9
Percentage of Participants With Mean S-K Values ≤ 5.1 mmol/L During Extended Dosing Phase Days 85 to 365 Primary · Study Days 85 to 365

Percentage of subjects with mean S-K values ≤ 5.1 mmol/L during Extended Dosing Phase - ITT Population

GroupValue95% CI
Percentage88.485.7 – 90.8

Adverse events — posted to ClinicalTrials.gov

Time frame: One year. Reporting threshold: 5%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

Acute Phase: ZS
Serious: 1/751 (0%)
Deaths: 0/751
Extended Dosing Phase: ZS
Serious: 161/746 (22%)
Deaths: 8/746

Serious adverse events (136 terms)

ReactionSystemAcute Phase: ZSExtended Dosing Phase: ZS
PneumoniaInfections and infestations
Cardiac failure congestiveCardiac disorders
Chest painGeneral disorders
OsteomyelitisInfections and infestations
Renal failure acuteRenal and urinary disorders
CellulitisInfections and infestations
Acute myocardial infarctionCardiac disorders
Acute respiratory failureRespiratory, thoracic and mediastinal disorders
DyspnoeaRespiratory, thoracic and mediastinal disorders
HypertensionVascular disorders
Cardiac failureCardiac disorders
Skin ulcerSkin and subcutaneous tissue disorders
Renal failure chronicRenal and urinary disorders
Urinary tract infectionInfections and infestations
HyperkalaemiaMetabolism and nutrition disorders
HypoglycaemiaMetabolism and nutrition disorders
Lobar pneumoniaInfections and infestations
Fluid overloadMetabolism and nutrition disorders
Angina unstableCardiac disorders
Chronic obstructive pulmonary diseaseRespiratory, thoracic and mediastinal disorders
Myocardial infarctionCardiac disorders
Pulmonary oedemaRespiratory, thoracic and mediastinal disorders
Atrial fibrillationCardiac disorders
Respiratory failureRespiratory, thoracic and mediastinal disorders
SepsisInfections and infestations
Other adverse events (7 terms — click to expand)

ReactionSystemAcute Phase: ZSExtended Dosing Phase: ZS
HypertensionVascular disorders
Oedema peripheralGeneral disorders
NauseaGastrointestinal disorders
Urinary tract infectionInfections and infestations
ConstipationGastrointestinal disorders
AnaemiaBlood and lymphatic system disorders
Upper respiratory infectionInfections and infestations

Most-reported serious reactions: Pneumonia, Cardiac failure congestive, Chest pain, Osteomyelitis, Renal failure acute, Cellulitis, Acute myocardial infarction, Acute respiratory failure.

Data from ClinicalTrials.gov NCT02163499 adverse events section.

Sponsor's own description

The Open-Label Maintenance Study contains an Acute Phase, in which subjects will be dosed with ZS 10 g three times daily (tid) for 24 to 72 hours, followed by a long-term Maintenance Phase.

Publications & conference data

8 peer-reviewed publications reference this trial (live from Europe PMC):

  1. Sodium Zirconium Cyclosilicate among Individuals with Hyperkalemia: A 12-Month Phase 3 Study.
    Spinowitz BS, Fishbane S, Pergola PE, Roger SD, et al · · 2019 · cited 151× · PMID 31110051 · DOI 10.2215/cjn.12651018
  2. Systematic Review and Meta-Analysis of Patiromer and Sodium Zirconium Cyclosilicate: A New Armamentarium for the Treatment of Hyperkalemia.
    Meaney CJ, Beccari MV, Yang Y, Zhao J. · · 2017 · cited 75× · PMID 28122118 · DOI 10.1002/phar.1906
  3. Long-term safety and efficacy of sodium zirconium cyclosilicate for hyperkalaemia in patients with mild/moderate versus severe/end-stage chronic kidney disease: comparative results from an open-label, Phase 3 study.
    Roger SD, Lavin PT, Lerma EV, McCullough PA, et al · · 2021 · cited 47× · PMID 32030422 · DOI 10.1093/ndt/gfz285
  4. Clinical utility of patiromer, sodium zirconium cyclosilicate, and sodium polystyrene sulfonate for the treatment of hyperkalemia: an evidence-based review.
    Beccari MV, Meaney CJ. · · 2017 · cited 46× · PMID 28356904 · DOI 10.2147/ce.s129555
  5. Pharmacological interventions for the acute management of hyperkalaemia in adults.
    Batterink J, Cessford TA, Taylor RA. · · 2015 · cited 21× · PMID 35658162 · DOI 10.1002/14651858.cd010344.pub2
  6. Cost effectiveness of sodium zirconium cyclosilicate for the treatment of hyperkalaemia in patients with CKD in Norway and Sweden.
    Kim K, Fagerström J, Chen G, Lagunova Z, et al · · 2022 · cited 13× · PMID 35953778 · DOI 10.1186/s12882-022-02903-7
  7. Recent advances in treatment of heart failure.
    Kitai T, Tang WW. · · 2015 · cited 11× · PMID 26918130 · DOI 10.12688/f1000research.7022.1
  8. Hyperkalaemia in Heart Failure.
    Ismail U, Sidhu K, Zieroth S. · · 2021 · cited 5× · PMID 34094588 · DOI 10.15420/cfr.2020.29

Verify or expand the search:

Other trials of Sodium Zirconium Cyclosilicate

Trials testing the same drug.

Other recruiting trials for Hyperkalemia

Currently open trials in the same condition.

Other ZS Pharma, Inc. trials

Trials by the same sponsor.

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Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT02163499.

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing