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NCT01892384

Safety and Tolerability of BI 409306 in Patients With Schizophrenia

Completed Phase 1 Results posted Last updated 25 April 2024
What this trial tests

Phase 1 trial testing Placebo in Schizophrenia in 40 participants. Completed in 5 December 2013.

Timeline
28 June 2013
Primary endpoint
5 December 2013
5 December 2013

Quick facts

Lead sponsorBoehringer Ingelheim
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationrandomized
Designparallel
Maskingdouble
Primary purposetreatment
Enrollment40
Start date28 June 2013
Primary completion5 December 2013
Estimated completion5 December 2013
Sites1 location across United States

Drugs / interventions tested

Conditions studied

Sponsor

Boehringer Ingelheim — full company profile →

Who can join

Adults 18 to 55, any sex, with Schizophrenia. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Number of Participants With Drug-related Adverse Events Primary · From first drug administration until 30 days after last drug administration, up to 44 days.

Number of participants with drug-related adverse events.

GroupValue95% CI
BI 409306 25mg1
BI 409306 50mg3
BI 409306 100mg2
Placebo3
Maximum Measured Concentration of BI 409306 in Plasma After Single Dose (Cmax) Secondary · 2 hours (h) before first drug administration and 10minutes (min), 20min, 30min, 45min, 1h, 1h 30min, 2h, 2h 30min, 3h, 4h, 6h, 8h, 10h, 12h and 14h after first drug administration

Maximum measured concentration of BI 409306 in plasma after single dose (Cmax) is presented.

GroupValue95% CI
BI 409306 25mg138± 91.9
BI 409306 50mg431± 73.3
BI 409306 100mg998± 106.0
Maximum Measured Concentration of BI 409306 in Plasma at Steady-state (Cmax,ss) Secondary · 2 hours (h) before drug administration and 10minutes (min), 20min, 30min, 45min, 1h, 1h 30min, 2h, 2h 30min, 3h, 4h, 6h, 8h, 10h, 12h, 14h, 24h, 48h and 72h after drug administration on day 14.

Maximum measured concentration of BI 409306 in plasma at steady-state (Cmax,ss) is presented.

GroupValue95% CI
BI 409306 25mg99.2± 86.8
BI 409306 50mg631± 90.9
BI 409306 100mg1290± 74.4
Time From Dosing to Maximum Measured Concentration of BI 409306 in Plasma After Single Dose (Tmax) Secondary · 2 hours (h) before first drug administration and 10minutes (min), 20min, 30min, 45min, 1h, 1h 30min, 2h, 2h 30min, 3h, 4h, 6h, 8h, 10h, 12h and 14h after first drug administration.

Time from dosing to maximum measured concentration of BI 409306 in plasma after single dose (tmax) is presented.

GroupValue95% CI
BI 409306 25mg0.6250.33 – 1.50
BI 409306 50mg0.6250.33 – 2.00
BI 409306 100mg0.7500.33 – 2.00
Time From Dosing to Maximum Measured Concentration of BI 409306 in Plasma at Steady-state (Tmax,ss) Secondary · 2 hours (h) before drug administration and 10minutes (min), 20min, 30min, 45min, 1h, 1h 30min, 2h, 2h 30min, 3h, 4h, 6h, 8h, 10h, 12h, 14h, 24h, 48h and 72h after drug administration on day 14.

Time from dosing to maximum measured concentration of BI 409306 in plasma at steady-state (tmax,ss) is presented.

GroupValue95% CI
BI 409306 25mg0.7500.33 – 1.00
BI 409306 50mg0.3330.33 – 1.50
BI 409306 100mg0.6250.33 – 1.50
Area Under the Concentration-time Curve of BI 409306 in Plasma Over the Time Interval From 0 Extrapolated to Infinity After a Single Dose (AUC0-infinity) Secondary · 2 hours (h) before first drug administration and 10minutes (min), 20min, 30min, 45min, 1h, 1h 30min, 2h, 2h 30min, 3h, 4h, 6h, 8h, 10h, 12h and 14h after first drug administration.

Area under the concentration-time curve of BI 409306 in plasma over the time interval from 0 extrapolated to infinity after a single dose (AUC0-infinity) is presented.

GroupValue95% CI
BI 409306 25mg217± 107.0
BI 409306 50mg770± 98.4
BI 409306 100mg2020± 108.0
Area Under the Concentration-time Curve of BI 409306 in Plasma at Steady State Over a Uniform Dosing Interval Tau (AUCtau,ss) Secondary · 2 hours (h) before drug administration and 10minutes (min), 20min, 30min, 45min, 1h, 1h 30min, 2h, 2h 30min, 3h, 4h, 6h, 8h, 10h, 12h, 14h, 24h, 48h and 72h after drug administration on day 14.

Area under the concentration-time curve of BI 409306 in plasma at steady state over a uniform dosing interval tau (AUCtau,ss) is presented.

GroupValue95% CI
BI 409306 25mg147± 112.0
BI 409306 50mg969± 104.0
BI 409306 100mg2280± 86.8

Adverse events — posted to ClinicalTrials.gov

Time frame: From first dose of study medication until 30 days after the last dose of study medication, up to 44 days.. Reporting threshold: 5%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

BI 409306 25mg
Serious: 0/10 (0%)
Deaths:
BI 409306 50mg
Serious: 0/10 (0%)
Deaths:
BI 409306 100mg
Serious: 0/10 (0%)
Deaths:
Placebo
Serious: 0/10 (0%)
Deaths:
Total.
Serious: 0/40 (0%)
Deaths:
Other adverse events (20 terms — click to expand)

ReactionSystemBI 409306 25mgBI 409306 50mgBI 409306 100mgPlaceboTotal.
Vision blurredEye disorders
PhotopsiaEye disorders
Visual impairmentEye disorders
ExcoriationInjury, poisoning and procedural complications
Musculoskeletal painMusculoskeletal and connective tissue disorders
HeadacheNervous system disorders
AgitationPsychiatric disorders
AnxietyPsychiatric disorders
Gastrooesophageal reflux diseaseGastrointestinal disorders
NauseaGastrointestinal disorders
ToothacheGastrointestinal disorders
VomitingGastrointestinal disorders
PainGeneral disorders
Pre-existing condition improvedGeneral disorders
FuruncleInfections and infestations
Tooth infectionInfections and infestations
Back painMusculoskeletal and connective tissue disorders
DizzinessNervous system disorders
TremorNervous system disorders
Visual field defectNervous system disorders

Data from ClinicalTrials.gov NCT01892384 adverse events section.

Sponsor's own description

The primary objective of the current study is to investigate the safety and tolerability of BI 409306 in schizophrenic patients following oral administration of multiple low, medium, and high doses over 14 days. A secondary objective is the exploration of the pharmacokinetics and pharmacodynamics of BI 409306 in schizophrenic patients.

Publications & conference data

2 peer-reviewed publications reference this trial (live from Europe PMC):

  1. Interventions for prodromal stage of psychosis.
    Bosnjak Kuharic D, Kekin I, Hew J, Rojnic Kuzman M, et al · · 2019 · cited 51× · PMID 31689359 · DOI 10.1002/14651858.cd012236.pub2
  2. A Phase IC Study Evaluating the Safety, Tolerability, Pharmacokinetics, and Cognitive Outcomes of BI 409306 in Patients with Mild-to-Moderate Schizophrenia.
    Brown D, Daniels K, Pichereau S, Sand M. · · 2018 · cited 6× · PMID 29177699 · DOI 10.1007/s40120-017-0085-5

Verify or expand the search:

Other trials of BI 409306

Trials testing the same drug.

Other recruiting trials for Schizophrenia

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Other Boehringer Ingelheim trials

Trials by the same sponsor.

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Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT01892384.

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing