PPAR-alpha — Drug Target
All drugs that target PPAR-alpha — marketed and clinical-stage. Includes 2 drug classes acting on this target.
Drug classes
Fibrate · Fatty acid ethyl ester
Phase 3 pipeline (1)
- bezafibrate (drug) · Assistance Publique - Hôpitaux de Paris · Fibrate · Cardiovascular
Bezafibrate is a fibric acid derivative that activates peroxisome proliferator-activated receptor alpha (PPAR-alpha), leading to increased lipolysis and decreased lipogenesis.
Phase 2 pipeline (1)
- Omega-3 fatty acid ethyl esters · Takeda · Fatty acid ethyl ester · Cardiovascular
Activates peroxisome proliferator-activated receptor alpha (PPAR-alpha)