Muscarinic acetylcholine receptor M4 — Drug Target
All drugs that target Muscarinic acetylcholine receptor M4 — marketed and clinical-stage. Includes 7 drug classes acting on this target.
Drug classes
Anticholinergic · Antiprotozoal · hyoscyamine · benzethonium · Antiemetic · Cholinergic Muscarinic Antagonist · Cholinergic Receptor Agonist
Marketed (9)
- Incruse Ellipta · Glaxo Grp England · Anticholinergic · Respiratory
Umeclidinium works by blocking the M4 muscarinic acetylcholine receptor to relax airway smooth muscle and improve breathing. - Pentam · Fresenius Kabi · Antiprotozoal · Metabolic
Pentamidine works by interfering with the reproduction of certain parasites, such as Pneumocystis jiroveci. - Pro-Banthine · Anticholinergic · Gastroenterology
- (-)-Atropine · University of Kansas Medical Center · hyoscyamine · Gastroenterology
- Benzetonium Chloride · benzethonium · Infectious Disease
- Cephadol · Antiemetic · Neuroscience
- Homatropin · Cholinergic Muscarinic Antagonist · Gastroenterology
- Salagen · Cholinergic Receptor Agonist · Oncology
- Methylrosaniline Chloride · Immunology