kappa opioid receptor — Drug Target

All drugs that target kappa opioid receptor — marketed and clinical-stage. Includes 5 drug classes acting on this target.

Drug classes

kappa opioid receptor antagonist · Opioid receptor antagonist · Kappa opioid receptor agonist · kappa opioid receptor agonist · opioid receptor antagonist

Phase 3 pipeline (2)

• Q8003 · QRxPharma Inc. · kappa opioid receptor antagonist · Psychiatry
  Q8003 is a selective inhibitor of the kappa opioid receptor.
• YM060 · Astellas Pharma Inc · kappa opioid receptor antagonist · Pain
  YM060 is a selective and potent kappa opioid receptor antagonist.

Phase 2 pipeline (6)

• Effentora® · Cephalon · Opioid receptor antagonist · Neurology
  A selective kappa opioid receptor antagonist.
• CNS 7056 · Paion UK Ltd. · Opioid receptor antagonist · Pain
  CNS 7056 is a kappa opioid receptor antagonist.
• ALC-2203-AC · Korea Arlico Pharm. Co., Ltd · Kappa opioid receptor agonist · Pain
  ALC-2203-AC is a selective and potent agonist of the kappa opioid receptor.
• Arm 1: CL-H1T · Charleston Laboratories, Inc · kappa opioid receptor agonist · Pain
  CL-H1T is a compound that targets the kappa opioid receptor.
• AC-203 · TWi Biotechnology, Inc. · kappa opioid receptor agonist · Pain
  AC-203 is a selective agonist of the kappa opioid receptor.
• A. CNS 7056 · Paion UK Ltd. · opioid receptor antagonist · Pain
  CNS 7056 is a kappa opioid receptor antagonist.