GnRH receptors — Drug Target

2 drugs 2 marketed

All drugs that target GnRH receptors — marketed and clinical-stage. Includes 2 drug classes acting on this target.

Drug classes

Gonadotropin Releasing Hormone Receptor Agonist · Progestin

Marketed (2)

Lupron · Accord Healthcare S.L.U. · Gonadotropin Releasing Hormone Receptor Agonist · Oncology
Leuprolide acetate, a long-acting GnRH analog, initially stimulates then suppresses pituitary gonadotropins, reducing gonadal steroid secretion.
Micronor · Johnson & Johnson · Progestin · Bone
ORIAHNN combines elagolix, which suppresses LH and FSH to reduce ovarian sex hormones, with estradiol and norethindrone acetate to mitigate side effects.