Endothelin-1 receptor — Drug Target

All drugs that target Endothelin-1 receptor — marketed and clinical-stage. Includes 3 drug classes acting on this target.

Drug classes

Endothelin Receptor Antagonist [EPC] · Endothelin Receptor Antagonist · Sulfonamide Antimicrobial

Marketed (5)

• Opsumit · AstraZeneca · Endothelin Receptor Antagonist [EPC] · Metabolic
  Opsumit works by blocking the action of endothelin-1, a protein that causes blood vessels to constrict and increase blood pressure.
• Pivlaz · Idorsia Pharmaceuticals Japan Ltd · Cardiovascular
• Tracleer · AstraZeneca · Endothelin Receptor Antagonist · Immunology
• Azo Gantrisin · Alra · Sulfonamide Antimicrobial · Immunology
• Letairis · Gilead Sciences · Endothelin Receptor Antagonist [EPC] · Cardiovascular