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Zidovudine (drug)
Zidovudine (drug) is a Nucleoside reverse transcriptase inhibitor (NRTI) Small molecule drug developed by Johann Wolfgang Goethe University Hospital. It is currently FDA-approved for HIV-1 infection, Prevention of maternal-fetal HIV transmission.
Zidovudine is a nucleoside reverse transcriptase inhibitor that blocks HIV replication by inhibiting the enzyme reverse transcriptase, preventing the virus from converting its RNA genome into DNA.
Zidovudine is a nucleoside reverse transcriptase inhibitor that blocks HIV replication by inhibiting the enzyme reverse transcriptase, preventing the virus from converting its RNA genome into DNA. Used for HIV-1 infection, Prevention of maternal-fetal HIV transmission.
At a glance
| Generic name | Zidovudine (drug) |
|---|---|
| Sponsor | Johann Wolfgang Goethe University Hospital |
| Drug class | Nucleoside reverse transcriptase inhibitor (NRTI) |
| Target | HIV reverse transcriptase |
| Modality | Small molecule |
| Therapeutic area | Infectious Disease / Virology |
| Phase | FDA-approved |
Mechanism of action
Zidovudine (AZT) is a thymidine analog that gets incorporated into the growing DNA chain during reverse transcription, causing chain termination and preventing HIV from replicating its genetic material. By inhibiting reverse transcriptase, it reduces viral load and slows disease progression in HIV-infected patients. It was the first antiretroviral drug approved for HIV treatment.
Approved indications
- HIV-1 infection
- Prevention of maternal-fetal HIV transmission
Common side effects
- Anemia
- Neutropenia
- Nausea
- Headache
- Fatigue
- Lactic acidosis
- Lipoatrophy
- Mitochondrial toxicity
Key clinical trials
- Virotherapy and Natural History Study of KHSV-Associated Multricentric Castleman s Disease With Correlates of Disease Activity (PHASE2)
- Study of Cobicistat-Boosted Atazanavir (ATV/co), Cobicistat-Boosted Darunavir (DRV/co) and Emtricitabine/Tenofovir Alafenamide (F/TAF) in Children With HIV (PHASE2, PHASE3)
- A Study to Provide Continued Access to Study Drug to Children and Adolescents Who Have Completed Clinical Studies Involving Gilead HIV Treatments (PHASE4)
- Natural History Study of the KSHV Inflammatory Cytokine Syndrome (KICS) (PHASE2)
- Belinostat Therapy With Zidovudine for Adult T-Cell Leukemia-Lymphoma (PHASE2)
- Effectiveness of Zidovudine vs. Zidovudine Plus Alpha Interferon vs. Interferon for Treatment of HIV
- Early Infant HIV Treatment in Botswana (PHASE2, PHASE3)
- Allogeneic Hematopoietic Cell Transplantation for Peripheral T Cell Lymphoma (PHASE2)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Zidovudine (drug) CI brief — competitive landscape report
- Zidovudine (drug) updates RSS · CI watch RSS
- Johann Wolfgang Goethe University Hospital portfolio CI
Frequently asked questions about Zidovudine (drug)
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Related
- Drug class: All Nucleoside reverse transcriptase inhibitor (NRTI) drugs
- Target: All drugs targeting HIV reverse transcriptase
- Manufacturer: Johann Wolfgang Goethe University Hospital — full pipeline
- Therapeutic area: All drugs in Infectious Disease / Virology
- Indication: Drugs for HIV-1 infection
- Indication: Drugs for Prevention of maternal-fetal HIV transmission
- Compare: Zidovudine (drug) vs similar drugs
- Pricing: Zidovudine (drug) cost, discount & access