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Xenetix-CT perfusion imaging

Guerbet · FDA-approved active Small molecule

Xenetix is an iodinated contrast medium that enhances visualization of blood perfusion in tissues during CT imaging by increasing radiodensity in vascular and tissue compartments.

Xenetix is an iodinated contrast medium that enhances visualization of blood perfusion in tissues during CT imaging by increasing radiodensity in vascular and tissue compartments. Used for CT perfusion imaging of the brain for acute stroke evaluation, CT perfusion imaging of the heart for myocardial ischemia assessment, CT perfusion imaging of solid organs for tumor characterization and tissue viability assessment.

At a glance

Generic nameXenetix-CT perfusion imaging
SponsorGuerbet
Drug classIodinated contrast medium
ModalitySmall molecule
Therapeutic areaDiagnostic Imaging
PhaseFDA-approved

Mechanism of action

Xenetix contains iopamidol, a non-ionic iodinated contrast agent that distributes through the vasculature and extracellular space. The iodine atoms attenuate X-rays, creating enhanced contrast between perfused and non-perfused tissues on CT scans. This allows quantitative assessment of regional blood flow and tissue perfusion in organs such as the brain, heart, and lungs.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results