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TAS-118 plus Oxaliplatin

Taiho Pharmaceutical Co., Ltd. · Phase 3 active Small molecule

TAS-118 is a thymidylate synthase inhibitor, and when combined with oxaliplatin, it targets rapidly dividing cancer cells.

TAS-118 is a thymidylate synthase inhibitor, and when combined with oxaliplatin, it targets rapidly dividing cancer cells. Used for Metastatic colorectal cancer.

At a glance

Generic nameTAS-118 plus Oxaliplatin
SponsorTaiho Pharmaceutical Co., Ltd.
Drug classThymidylate synthase inhibitor
TargetThymidylate synthase
ModalitySmall molecule
Therapeutic areaOncology
PhasePhase 3

Mechanism of action

TAS-118 works by inhibiting thymidylate synthase, an enzyme involved in DNA synthesis. This leads to the inhibition of cancer cell growth and proliferation. When combined with oxaliplatin, a platinum-based chemotherapy drug, the combination targets rapidly dividing cancer cells, leading to cell death.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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