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Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin
Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin is a Antimalarial Small molecule drug developed by London School of Hygiene and Tropical Medicine. It is currently in Phase 3 development for Treatment of uncomplicated malaria, Prevention of malaria in areas with high transmission.
Sulphadoxine acts as a sulfonamide antibacterial agent, inhibiting dihydropteroate synthase, while pyrimethamine inhibits dihydrofolate reductase, and amodiaquine is a 4-aminoquinoline antimalarial that targets the malaria parasite's heme detoxification pathway. Azithromycin is a macrolide antibiotic that inhibits protein synthesis in bacteria.
Sulphadoxine acts as a sulfonamide antibacterial agent, inhibiting dihydropteroate synthase, while pyrimethamine inhibits dihydrofolate reductase, and amodiaquine is a 4-aminoquinoline antimalarial that targets the malaria parasite's heme detoxification pathway. Azithromycin is a macrolide antibiotic that inhibits protein synthesis in bacteria. Used for Treatment of uncomplicated malaria, Prevention of malaria in areas with high transmission.
At a glance
| Generic name | Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin |
|---|---|
| Sponsor | London School of Hygiene and Tropical Medicine |
| Drug class | Antimalarial |
| Target | Dihydropteroate synthase, Dihydrofolate reductase, Heme detoxification pathway |
| Modality | Small molecule |
| Therapeutic area | Infectious Diseases |
| Phase | Phase 3 |
Mechanism of action
Sulphadoxine and pyrimethamine are a combination of two drugs that work synergistically to treat malaria. Sulphadoxine inhibits the growth of the malaria parasite by interfering with its ability to synthesize folic acid, while pyrimethamine targets the parasite's dihydrofolate reductase enzyme. Amodiaquine is another antimalarial drug that targets the parasite's heme detoxification pathway. Azithromycin, on the other hand, is a broad-spectrum antibiotic that targets a wide range of bacteria by inhibiting protein synthesis.
Approved indications
- Treatment of uncomplicated malaria
- Prevention of malaria in areas with high transmission
Common side effects
- Nausea
- Vomiting
- Diarrhea
- Abdominal pain
- Headache
Key clinical trials
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin CI brief — competitive landscape report
- Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin updates RSS · CI watch RSS
- London School of Hygiene and Tropical Medicine portfolio CI
Frequently asked questions about Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin
What is Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin?
How does Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin work?
What is Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin used for?
Who makes Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin?
What drug class is Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin in?
What development phase is Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin in?
What are the side effects of Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin?
What does Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin target?
Related
- Drug class: All Antimalarial drugs
- Target: All drugs targeting Dihydropteroate synthase, Dihydrofolate reductase, Heme detoxification pathway
- Manufacturer: London School of Hygiene and Tropical Medicine — full pipeline
- Therapeutic area: All drugs in Infectious Diseases
- Indication: Drugs for Treatment of uncomplicated malaria
- Indication: Drugs for Prevention of malaria in areas with high transmission
- Compare: Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin vs similar drugs
- Pricing: Sulphadoxine-Pyrimethamine+ Amodiaquine+ Azithromycin cost, discount & access